PMC:7461420 / 69854-70195
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T269 | 335-340 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T332 | 144-148 | Disease | denotes | SARS | http://purl.obolibrary.org/obo/MONDO_0005091 |
T333 | 307-311 | Disease | denotes | SARS | http://purl.obolibrary.org/obo/MONDO_0005091 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T845 | 163-164 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T846 | 203-204 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T847 | 267-275 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T848 | 327-340 | http://purl.obolibrary.org/obo/CLO_0051719 | denotes | Vero E6 cells |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T81382 | 257-266 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
2179 | 155-159 | Gene | denotes | Mpro | Gene:8673700 |
2180 | 45-49 | Gene | denotes | Mpro | Gene:8673700 |
2185 | 144-152 | Species | denotes | SARS‐CoV | Tax:694009 |
2186 | 13-20 | Chemical | denotes | (R)‐123 | |
2187 | 126-133 | Chemical | denotes | (R)‐123 | |
2188 | 237-244 | Chemical | denotes | (R)‐123 | |
2189 | 294-302 | Disease | denotes | infected | MESH:D007239 |
2190 | 307-331 | Disease | denotes | SARS‐CoV‐1 infected Vero | MESH:C000657245 |
2191 | 332-334 | CellLine | denotes | E6 | CVCL:4582 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T606 | 0-341 | Sentence | denotes | Indeed, only (R)‐123 was able to inhibit the Mpro enzyme with an IC50 value of 1.5 µM, while the (S)‐enantiomer was inactive. (R)‐123 inhibited SARS‐CoV‐1 Mpro in a competitive manner (K i, 1.6 µM) with a noncovalent mode of inhibition. (R)‐123 also showed antiviral activity (12.9 µM) in mock infected and SARS‐CoV‐1 infected Vero E6 cells. |