| Id |
Subject |
Object |
Predicate |
Lexical cue |
| T118 |
0-216 |
Sentence |
denotes |
To improve the solubility characteristics of inhibitors incorporating the lipophilic 2,6-dichlorobenzoate, a limited set of inhibitors containing smaller or more polar amine capping fragments were prepared (Table 2). |
| T119 |
217-304 |
Sentence |
denotes |
Replacement of the 4-methoxy indole cap present in 22 with a benzimidazole provided 31. |
| T120 |
305-416 |
Sentence |
denotes |
This inhibitor displayed potent irreversible inhibition kinetics but did not improve solubility compared to 22. |
| T121 |
417-574 |
Sentence |
denotes |
Reduction in the size of the P2 capping element as represented by 29 and 30 provided derivatives that possessed weak reversible SARS CoV-1 3CLpro inhibition. |
