Id |
Subject |
Object |
Predicate |
Lexical cue |
T581 |
0-70 |
Sentence |
denotes |
Zhou et al. extended the SAR studies for further activity improvement. |
T582 |
71-156 |
Sentence |
denotes |
Compound 108 bearing carboxamide showed the best SARS‐CoV‐1 Mpro inhibitory activity. |
T583 |
157-247 |
Sentence |
denotes |
However, this derivative did not bind covalently to the Cys145 residue of the active site. |
T584 |
248-385 |
Sentence |
denotes |
177 Further structural investigations at the carboxamide of 108 with a variety of substituted sulfonamides did not improve the activity. |
T585 |
386-443 |
Sentence |
denotes |
Compound 109 was the best one of that series (Figure 28). |
T586 |
444-447 |
Sentence |
denotes |
178 |