PMC:7600245 / 29542-30498
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T122 | 147-152 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T123 | 760-767 | Body_part | denotes | protein | http://purl.org/sig/ont/fma/fma67257 |
T124 | 822-825 | Body_part | denotes | HIV | http://purl.org/sig/ont/fma/fma278683 |
T125 | 899-902 | Body_part | denotes | HIV | http://purl.org/sig/ont/fma/fma278683 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T110 | 119-127 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T111 | 400-408 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T112 | 668-676 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T113 | 947-955 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T271 | 102-110 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T272 | 130-135 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T273 | 139-152 | http://purl.obolibrary.org/obo/CLO_0051719 | denotes | Vero E6 cells |
T274 | 192-197 | http://purl.obolibrary.org/obo/CLO_0007488 | denotes | M [85 |
T275 | 324-330 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | active |
T276 | 383-391 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T277 | 473-479 | http://purl.obolibrary.org/obo/NCBITaxon_33208 | denotes | animal |
T278 | 745-749 | http://purl.obolibrary.org/obo/CLO_0001649 | denotes | a C2 |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T418 | 24-33 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T419 | 69-78 | Chemical | denotes | Lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T420 | 92-101 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T421 | 247-256 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T422 | 354-363 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T423 | 590-609 | Chemical | denotes | lopinavir/ritonavir | http://purl.obolibrary.org/obo/CHEBI_145924 |
T424 | 590-599 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T425 | 600-609 | Chemical | denotes | ritonavir | http://purl.obolibrary.org/obo/CHEBI_45409 |
T426 | 625-634 | Chemical | denotes | ribavirin | http://purl.obolibrary.org/obo/CHEBI_63580 |
T427 | 747-749 | Chemical | denotes | C2 | http://purl.obolibrary.org/obo/CHEBI_30083 |
T428 | 760-767 | Chemical | denotes | protein | http://purl.obolibrary.org/obo/CHEBI_36080 |
T429 | 804-813 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T430 | 828-847 | Chemical | denotes | protease inhibitors | http://purl.obolibrary.org/obo/CHEBI_37670|http://purl.obolibrary.org/obo/CHEBI_60258 |
T432 | 837-847 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
T433 | 905-914 | Chemical | denotes | aspartate | http://purl.obolibrary.org/obo/CHEBI_132943|http://purl.obolibrary.org/obo/CHEBI_29995|http://purl.obolibrary.org/obo/CHEBI_72314 |
T436 | 915-934 | Chemical | denotes | protease inhibitors | http://purl.obolibrary.org/obo/CHEBI_37670|http://purl.obolibrary.org/obo/CHEBI_60258 |
T438 | 924-934 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T217 | 0-68 | Sentence | denotes | The rationale for using lopinavir is attributed to multiple studies. |
T218 | 69-199 | Sentence | denotes | Lopinavir exhibited an antiviral activity against SARS-CoV-2 virus in Vero E6 cells with an estimated EC50 value of 26.63 μM [85]. |
T219 | 200-344 | Sentence | denotes | Computational studies have also suggested that lopinavir may inhibit the viral main protease Mpro, perhaps by targeting its active site [86,87]. |
T220 | 345-435 | Sentence | denotes | Earlier, lopinavir exhibited in vitro activity against SARS-CoV-1 and MERS-CoV [88,89,90]. |
T221 | 436-526 | Sentence | denotes | It also showed beneficial effects in animal studies for the treatment of MERS-CoV [91,92]. |
T222 | 527-688 | Sentence | denotes | Furthermore, there is an evidence of some clinical benefit for lopinavir/ritonavir when used with ribavirin and/or INFs against MERS-CoV and SARS-CoV [88,93,94]. |
T223 | 689-848 | Sentence | denotes | Yet, coronavirus proteases, including Mpro, do not have a C2-symmetric protein architecture which is the target of lopinavir and all HIV-1 protease inhibitors. |
T224 | 849-956 | Sentence | denotes | This subsequently sheds doubts on the prospect of HIV-1 aspartate protease inhibitors in treating COVID-19. |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
846 | 293-297 | Gene | denotes | Mpro | Gene:8673700 |
847 | 727-731 | Gene | denotes | Mpro | Gene:8673700 |
848 | 119-129 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
849 | 400-408 | Species | denotes | SARS-CoV | Tax:694009 |
850 | 415-423 | Species | denotes | MERS-CoV | Tax:1335626 |
851 | 509-517 | Species | denotes | MERS-CoV | Tax:1335626 |
852 | 655-663 | Species | denotes | MERS-CoV | Tax:1335626 |
853 | 668-676 | Species | denotes | SARS-CoV | Tax:694009 |
854 | 694-705 | Species | denotes | coronavirus | Tax:11118 |
855 | 822-827 | Species | denotes | HIV-1 | Tax:11676 |
856 | 899-904 | Species | denotes | HIV-1 | Tax:11676 |
857 | 24-33 | Chemical | denotes | lopinavir | MESH:D061466 |
858 | 69-78 | Chemical | denotes | Lopinavir | MESH:D061466 |
859 | 247-256 | Chemical | denotes | lopinavir | MESH:D061466 |
860 | 354-363 | Chemical | denotes | lopinavir | MESH:D061466 |
861 | 590-609 | Chemical | denotes | lopinavir/ritonavir | MESH:C558899 |
862 | 625-634 | Chemical | denotes | ribavirin | MESH:D012254 |
863 | 804-813 | Chemical | denotes | lopinavir | MESH:D061466 |
864 | 947-955 | Disease | denotes | COVID-19 | MESH:C000657245 |
865 | 139-146 | CellLine | denotes | Vero E6 | CVCL:0574 |