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PMC:7600245 / 25077-26455
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T101 | 41-47 | Body_part | denotes | purine | http://purl.org/sig/ont/fma/fma82772 |
T102 | 48-58 | Body_part | denotes | nucleotide | http://purl.org/sig/ont/fma/fma82740 |
T103 | 159-162 | Body_part | denotes | RNA | http://purl.org/sig/ont/fma/fma67095 |
T104 | 589-598 | Body_part | denotes | histidine | http://purl.org/sig/ont/fma/fma82755 |
T105 | 605-615 | Body_part | denotes | nucleotide | http://purl.org/sig/ont/fma/fma82740 |
T106 | 624-631 | Body_part | denotes | protein | http://purl.org/sig/ont/fma/fma67257 |
T107 | 807-814 | Body_part | denotes | protein | http://purl.org/sig/ont/fma/fma67257 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T97 | 1156-1165 | Disease | denotes | cirrhosis | http://purl.obolibrary.org/obo/MONDO_0005155 |
T98 | 1337-1345 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T229 | 33-39 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | active |
T230 | 86-89 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T231 | 110-118 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T232 | 163-170 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | viruses |
T233 | 182-187 | http://purl.obolibrary.org/obo/NCBITaxon_9606 | denotes | human |
T234 | 231-232 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T235 | 395-405 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activation |
T236 | 458-463 | http://purl.obolibrary.org/obo/NCBITaxon_9606 | denotes | human |
T237 | 507-508 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | A |
T238 | 948-954 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | active |
T239 | 1071-1079 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T240 | 1213-1214 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T338 | 41-58 | Chemical | denotes | purine nucleotide | http://purl.obolibrary.org/obo/CHEBI_26395 |
T339 | 41-47 | Chemical | denotes | purine | http://purl.obolibrary.org/obo/CHEBI_35584 |
T340 | 48-58 | Chemical | denotes | nucleotide | http://purl.obolibrary.org/obo/CHEBI_36976 |
T341 | 59-66 | Chemical | denotes | prodrug | http://purl.obolibrary.org/obo/CHEBI_50266 |
T342 | 75-77 | Chemical | denotes | S3 | http://purl.obolibrary.org/obo/CHEBI_29388 |
T343 | 100-109 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T344 | 240-249 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T345 | 308-320 | Chemical | denotes | sulfate salt | http://purl.obolibrary.org/obo/CHEBI_35175 |
T346 | 308-315 | Chemical | denotes | sulfate | http://purl.obolibrary.org/obo/CHEBI_16189 |
T347 | 316-320 | Chemical | denotes | salt | http://purl.obolibrary.org/obo/CHEBI_24866|http://purl.obolibrary.org/obo/CHEBI_26710 |
T349 | 326-330 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T350 | 531-539 | Chemical | denotes | L-alanyl | http://purl.obolibrary.org/obo/CHEBI_32433|http://purl.obolibrary.org/obo/CHEBI_46217 |
T352 | 533-539 | Chemical | denotes | alanyl | http://purl.obolibrary.org/obo/CHEBI_22280|http://purl.obolibrary.org/obo/CHEBI_32441 |
T354 | 589-598 | Chemical | denotes | histidine | http://purl.obolibrary.org/obo/CHEBI_27570 |
T355 | 605-615 | Chemical | denotes | nucleotide | http://purl.obolibrary.org/obo/CHEBI_36976 |
T356 | 624-631 | Chemical | denotes | protein | http://purl.obolibrary.org/obo/CHEBI_36080 |
T357 | 708-718 | Chemical | denotes | metabolite | http://purl.obolibrary.org/obo/CHEBI_25212 |
T358 | 762-771 | Chemical | denotes | guanosine | http://purl.obolibrary.org/obo/CHEBI_16750 |
T359 | 782-791 | Chemical | denotes | adenosine | http://purl.obolibrary.org/obo/CHEBI_16335 |
T360 | 807-814 | Chemical | denotes | protein | http://purl.obolibrary.org/obo/CHEBI_36080 |
T361 | 886-908 | Chemical | denotes | nucleoside diphosphate | http://purl.obolibrary.org/obo/CHEBI_16862 |
T362 | 886-896 | Chemical | denotes | nucleoside | http://purl.obolibrary.org/obo/CHEBI_33838 |
T363 | 897-908 | Chemical | denotes | diphosphate | http://purl.obolibrary.org/obo/CHEBI_18361|http://purl.obolibrary.org/obo/CHEBI_33019 |
T365 | 970-981 | Chemical | denotes | diphosphate | http://purl.obolibrary.org/obo/CHEBI_18361|http://purl.obolibrary.org/obo/CHEBI_33019 |
T367 | 1017-1019 | Chemical | denotes | S3 | http://purl.obolibrary.org/obo/CHEBI_29388 |
T368 | 1061-1070 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T369 | 1176-1180 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
LitCovid-PD-GO-BP
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T45 | 677-686 | http://purl.obolibrary.org/obo/GO_0009058 | denotes | formation |
LitCovid-PD-HP
Id | Subject | Object | Predicate | Lexical cue | hp_id |
---|---|---|---|---|---|
T15 | 1156-1165 | Phenotype | denotes | cirrhosis | http://purl.obolibrary.org/obo/HP_0001394 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T183 | 0-224 | Sentence | denotes | It is an investigational, orally active, purine nucleotide prodrug (Figure S3), which has exhibited antiviral activity against many single-stranded, enveloped RNA viruses, including human flaviviruses and coronaviruses [77]. |
T184 | 225-269 | Sentence | denotes | It is a potent inhibitor of viral RdRp [78]. |
T185 | 270-412 | Sentence | denotes | Following oral administration as hemi-sulfate salt, the drug gets converted to the monophosphate form via multiple metabolic activation steps. |
T186 | 413-553 | Sentence | denotes | The first step is catalyzed by the action of human carboxylesterase 1 (CES1) and/or cathepsin A (CatA) to produce the L-alanyl intermediate. |
T187 | 554-719 | Sentence | denotes | Spontaneous hydrolysis followed by histidine triad nucleotide-binding protein 1 (HINT1)-mediated hydrolysis results in the formation of the monophosphate metabolite. |
T188 | 720-1026 | Sentence | denotes | Then, the monophosphate is transformed to guanosine analog by adenosine deaminase like protein 1 (ADALP1) and further phosphorylated by guanylate kinase 1 (GUK1) and nucleoside diphosphate kinase (NDPK) to the pharmacologically active form of AT-527 diphosphate (also reported as AT-9010) (Figure S3) [78]. |
T189 | 1027-1171 | Sentence | denotes | The safety, pharmacokinetics, and antiviral activity of AT-527 was earlier established in HCV-infected subjects with and without cirrhosis [79]. |
T190 | 1172-1378 | Sentence | denotes | The drug is currently being evaluated in a phase 2 double-blind, randomized, placebo-controlled study to determine its efficacy and safety in patients with moderate COVID-19 symptoms (NCT04396106; n = 190). |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
707 | 259-263 | Gene | denotes | RdRp | Gene:43740578 |
708 | 464-482 | Gene | denotes | carboxylesterase 1 | Gene:1066 |
709 | 484-488 | Gene | denotes | CES1 | Gene:1066 |
710 | 497-508 | Gene | denotes | cathepsin A | Gene:5476 |
711 | 510-514 | Gene | denotes | CatA | Gene:5476 |
712 | 589-633 | Gene | denotes | histidine triad nucleotide-binding protein 1 | Gene:3094 |
713 | 635-640 | Gene | denotes | HINT1 | Gene:3094 |
714 | 856-874 | Gene | denotes | guanylate kinase 1 | Gene:2987 |
715 | 876-880 | Gene | denotes | GUK1 | Gene:2987 |
716 | 886-915 | Gene | denotes | nucleoside diphosphate kinase | Gene:129607 |
717 | 917-921 | Gene | denotes | NDPK | Gene:129607 |
718 | 182-187 | Species | denotes | human | Tax:9606 |
719 | 205-218 | Species | denotes | coronaviruses | Tax:11118 |
720 | 458-463 | Species | denotes | human | Tax:9606 |
721 | 1314-1322 | Species | denotes | patients | Tax:9606 |
722 | 41-58 | Chemical | denotes | purine nucleotide | MESH:D011685 |
723 | 303-320 | Chemical | denotes | hemi-sulfate salt | |
724 | 353-366 | Chemical | denotes | monophosphate | |
725 | 531-539 | Chemical | denotes | L-alanyl | |
726 | 694-707 | Chemical | denotes | monophosphate | |
727 | 730-743 | Chemical | denotes | monophosphate | |
728 | 762-771 | Chemical | denotes | guanosine | MESH:D006151 |
729 | 782-791 | Chemical | denotes | adenosine | MESH:D000241 |
730 | 970-981 | Chemical | denotes | diphosphate | MESH:D011756 |
731 | 1117-1129 | Disease | denotes | HCV-infected | MESH:D006526 |
732 | 1156-1165 | Disease | denotes | cirrhosis | MESH:D005355 |
733 | 1337-1345 | Disease | denotes | COVID-19 | MESH:C000657245 |