PMC:7128678 / 9990-11094
Annnotations
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
301 | 796-802 | Gene | denotes | CLQ-OH | |
302 | 705-723 | Chemical | denotes | hydroxychloroquine | MESH:D006886 |
303 | 725-731 | Chemical | denotes | CLQ-OH | |
304 | 750-762 | Chemical | denotes | sialic acids | MESH:D012794 |
305 | 812-846 | Chemical | denotes | N-acetyl-9-O-acetylneuraminic acid | MESH:C025676 |
306 | 848-855 | Chemical | denotes | 9-O-SIA | |
307 | 946-952 | Chemical | denotes | CLQ-OH | |
308 | 1014-1020 | Chemical | denotes | CLQ-OH | |
309 | 1087-1095 | Chemical | denotes | hydrogen | MESH:D006859 |
316 | 6-12 | Chemical | denotes | CLQ-OH | |
317 | 113-119 | Chemical | denotes | CLQ-OH | |
318 | 310-316 | Chemical | denotes | CLQ-OH | |
319 | 350-361 | Chemical | denotes | sialic acid | MESH:D019158 |
320 | 389-397 | Chemical | denotes | hydrogen | MESH:D006859 |
321 | 430-438 | Chemical | denotes | hydrogen | MESH:D006859 |
LitCovid-PMC-OGER-BB
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T230 | 91-98 | GO:0032991 | denotes | complex |
T231 | 298-300 | CHEBI:46882;CHEBI:46882 | denotes | OH |
T232 | 301-306 | CHEBI:24433;CHEBI:24433 | denotes | group |
T233 | 350-361 | CHEBI:26667;CHEBI:26667 | denotes | sialic acid |
T234 | 567-574 | GO:0032991 | denotes | complex |
T235 | 705-723 | CHEBI:5801;DG_20;CHEBI:5801 | denotes | hydroxychloroquine |
T236 | 750-762 | CHEBI:26667;CHEBI:26667 | denotes | sialic acids |
T237 | 812-846 | CHEBI:21500;CHEBI:21500 | denotes | N-acetyl-9-O-acetylneuraminic acid |
T238 | 884-891 | GO:0032991 | denotes | complex |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T64 | 17-23 | http://purl.obolibrary.org/obo/UBERON_0000473 | denotes | tested |
T65 | 179-180 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T66 | 181-182 | http://purl.obolibrary.org/obo/CLO_0001021 | denotes | b |
T67 | 387-388 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T68 | 661-663 | http://purl.obolibrary.org/obo/CLO_0053799 | denotes | 45 |
T69 | 765-766 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T70 | 767-768 | http://purl.obolibrary.org/obo/CLO_0001021 | denotes | b |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T167 | 301-306 | Chemical | denotes | group | http://purl.obolibrary.org/obo/CHEBI_24433 |
T168 | 350-361 | Chemical | denotes | sialic acid | http://purl.obolibrary.org/obo/CHEBI_26667 |
T169 | 357-361 | Chemical | denotes | acid | http://purl.obolibrary.org/obo/CHEBI_37527 |
T170 | 389-397 | Chemical | denotes | hydrogen | http://purl.obolibrary.org/obo/CHEBI_49637 |
T171 | 430-438 | Chemical | denotes | hydrogen | http://purl.obolibrary.org/obo/CHEBI_49637 |
T172 | 705-723 | Chemical | denotes | hydroxychloroquine | http://purl.obolibrary.org/obo/CHEBI_5801 |
T173 | 750-762 | Chemical | denotes | sialic acids | http://purl.obolibrary.org/obo/CHEBI_26667 |
T174 | 757-762 | Chemical | denotes | acids | http://purl.obolibrary.org/obo/CHEBI_37527 |
T175 | 812-846 | Chemical | denotes | N-acetyl-9-O-acetylneuraminic acid | http://purl.obolibrary.org/obo/CHEBI_21500 |
T176 | 814-820 | Chemical | denotes | acetyl | http://purl.obolibrary.org/obo/CHEBI_40574|http://purl.obolibrary.org/obo/CHEBI_46887 |
T178 | 842-846 | Chemical | denotes | acid | http://purl.obolibrary.org/obo/CHEBI_37527 |
T179 | 1087-1095 | Chemical | denotes | hydrogen | http://purl.obolibrary.org/obo/CHEBI_49637 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T76 | 0-86 | Sentence | denotes | Next, CLQ-OH was tested to assess whether it could, as CLQ, bind to 9-O-SIA (Fig. 3 ). |
T77 | 87-278 | Sentence | denotes | The complex obtained with CLQ-OH was very similar to that obtained with CLQ [compare Fig. 3(a,b) with Fig. 2(e,f), although several conformational adjustments occurred during the simulations. |
T78 | 279-415 | Sentence | denotes | Interestingly, the OH group of CLQ-OH reinforced the binding of CLQ to sialic acid through establishment of a hydrogen bond Fig. 3(c,d). |
T79 | 416-674 | Sentence | denotes | Overall, this hydrogen bond compensated for the slight loss of energy caused by the conformational rearrangement, and the energy of interaction of the complex was estimated to be -46 kJ.mol−1, which is very close to the value obtained for CLQ (-45 kJ.mol−1). |
T80 | 675-857 | Sentence | denotes | Fig. 3 Molecular modelling of hydroxychloroquine (CLQ-OH) interaction with sialic acids. (a,b) Surface representation of CLQ-OH bound to N-acetyl-9-O-acetylneuraminic acid (9-O-SIA). |
T81 | 858-902 | Sentence | denotes | Two opposite views of the complex are shown. |
T82 | 903-1104 | Sentence | denotes | Note the geometric complementarity between CLQ-OH (in blue) and 9-O-SIA (in red). (c,d) Molecular mechanism of CLQ-OH binding to 9-O-SIA: combination of electrostatic interactions and hydrogen bonding. |