PubMed:29194348
Annnotations
GoldHamster
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 2-13 | D005959 | denotes | Glucosidase |
T10 | 18-49 | P20417 | denotes | Protein Tyrosine Phosphatase 1B |
T11 | 18-49 | P35821 | denotes | Protein Tyrosine Phosphatase 1B |
T12 | 18-49 | P18031 | denotes | Protein Tyrosine Phosphatase 1B |
T14 | 18-49 | O13016 | denotes | Protein Tyrosine Phosphatase 1B |
T15 | 18-49 | PR:000013448 | denotes | Protein Tyrosine Phosphatase 1B |
T13 | 18-49 | D054562 | denotes | Protein Tyrosine Phosphatase 1B |
T17 | 26-34 | 10962 | denotes | Tyrosine |
T21 | 26-34 | SO:0001446 | denotes | Tyrosine |
T23 | 35-46 | GO:0016791 | denotes | Phosphatase |
T26 | 111-134 | 127450 | denotes | Sargassum serratifolium |
T27 | 171-183 | D000459 | denotes | Phaeophyceae |
T28 | 460-471 | CHEBI:22586 | denotes | antioxidant |
T33 | 630-637 | SO:0000104 | denotes | protein |
T29 | 630-637 | GO:0003675 | denotes | protein |
T41 | 630-661 | P20417 | denotes | protein tyrosine phosphatase 1B |
T42 | 630-661 | P35821 | denotes | protein tyrosine phosphatase 1B |
T43 | 630-661 | P18031 | denotes | protein tyrosine phosphatase 1B |
T45 | 630-661 | O13016 | denotes | protein tyrosine phosphatase 1B |
T46 | 630-661 | PR:000013448 | denotes | protein tyrosine phosphatase 1B |
T44 | 630-661 | D054562 | denotes | protein tyrosine phosphatase 1B |
T48 | 638-646 | 10962 | denotes | tyrosine |
T52 | 638-646 | SO:0001446 | denotes | tyrosine |
T54 | 647-658 | GO:0016791 | denotes | phosphatase |
T79 | 663-666 | CHEBI:52242 | denotes | PTP |
T93 | 663-668 | P20417 | denotes | PTP1B |
T94 | 663-668 | P35821 | denotes | PTP1B |
T95 | 663-668 | PR:O13016 | denotes | PTP1B |
T96 | 663-668 | P18031 | denotes | PTP1B |
T97 | 663-668 | O13016 | denotes | PTP1B |
T98 | 663-668 | PR:000013448 | denotes | PTP1B |
T99 | 663-668 | PR:P18031 | denotes | PTP1B |
T100 | 673-684 | D005959 | denotes | glucosidase |
T101 | 690-694 | CHEBI:29330 | denotes | ONOO |
T102 | 713-722 | MOP:0000556 | denotes | nitration |
T126 | 789-792 | CHEBI:52242 | denotes | PTP |
T140 | 789-794 | P20417 | denotes | PTP1B |
T141 | 789-794 | P35821 | denotes | PTP1B |
T142 | 789-794 | PR:O13016 | denotes | PTP1B |
T143 | 789-794 | P18031 | denotes | PTP1B |
T144 | 789-794 | O13016 | denotes | PTP1B |
T145 | 789-794 | PR:000013448 | denotes | PTP1B |
T146 | 789-794 | PR:P18031 | denotes | PTP1B |
T147 | 801-812 | D005959 | denotes | glucosidase |
T172 | 875-878 | CHEBI:52242 | denotes | PTP |
T186 | 875-880 | P20417 | denotes | PTP1B |
T187 | 875-880 | P35821 | denotes | PTP1B |
T188 | 875-880 | PR:O13016 | denotes | PTP1B |
T189 | 875-880 | P18031 | denotes | PTP1B |
T190 | 875-880 | O13016 | denotes | PTP1B |
T191 | 875-880 | PR:000013448 | denotes | PTP1B |
T192 | 875-880 | PR:P18031 | denotes | PTP1B |
T193 | 887-898 | D005959 | denotes | glucosidase |
T194 | 984-1006 | C528847 | denotes | sargahydroquinoic acid |
T195 | 984-1006 | C528847 | denotes | sargahydroquinoic acid |
T197 | 1008-1022 | C503204 | denotes | sargachromenol |
T198 | 1008-1022 | C503204 | denotes | sargachromenol |
T199 | 1027-1044 | C477718 | denotes | sargaquinoic acid |
T200 | 1027-1044 | C477718 | denotes | sargaquinoic acid |
T202 | 1076-1084 | CHEBI:29021 | denotes | n-hexane |
T203 | 1076-1084 | C026385 | denotes | n-hexane |
T204 | 1076-1084 | C026385 | denotes | n-hexane |
T229 | 1193-1196 | CHEBI:52242 | denotes | PTP |
T243 | 1193-1198 | P20417 | denotes | PTP1B |
T244 | 1193-1198 | P35821 | denotes | PTP1B |
T245 | 1193-1198 | PR:O13016 | denotes | PTP1B |
T246 | 1193-1198 | P18031 | denotes | PTP1B |
T247 | 1193-1198 | O13016 | denotes | PTP1B |
T248 | 1193-1198 | PR:000013448 | denotes | PTP1B |
T249 | 1193-1198 | PR:P18031 | denotes | PTP1B |
T250 | 1241-1255 | C503204 | denotes | sargachromenol |
T251 | 1241-1255 | C503204 | denotes | sargachromenol |
T252 | 1260-1277 | C477718 | denotes | sargaquinoic acid |
T253 | 1260-1277 | C477718 | denotes | sargaquinoic acid |
T255 | 1330-1341 | D005959 | denotes | glucosidase |
T279 | 1421-1424 | CHEBI:52242 | denotes | PTP |
T293 | 1421-1426 | P20417 | denotes | PTP1B |
T294 | 1421-1426 | P35821 | denotes | PTP1B |
T295 | 1421-1426 | PR:O13016 | denotes | PTP1B |
T296 | 1421-1426 | P18031 | denotes | PTP1B |
T297 | 1421-1426 | O13016 | denotes | PTP1B |
T298 | 1421-1426 | PR:000013448 | denotes | PTP1B |
T299 | 1421-1426 | PR:P18031 | denotes | PTP1B |
T300 | 1425-1433 | P10773 | denotes | B enzyme |
T301 | 1446-1468 | C528847 | denotes | sargahydroquinoic acid |
T302 | 1446-1468 | C528847 | denotes | sargahydroquinoic acid |
T304 | 1473-1490 | C477718 | denotes | sargaquinoic acid |
T305 | 1473-1490 | C477718 | denotes | sargaquinoic acid |
T307 | 1529-1543 | C503204 | denotes | sargachromenol |
T308 | 1529-1543 | C503204 | denotes | sargachromenol |
T309 | 1638-1642 | CHEBI:29330 | denotes | ONOO |
T310 | 1661-1670 | MOP:0000556 | denotes | nitration |
T311 | 1738-1745 | SO:0100018 | denotes | binding |
T312 | 1738-1745 | SO:0001091 | denotes | binding |
T313 | 1738-1745 | GO:0005488 | denotes | binding |
T314 | 1794-1801 | SO:0100018 | denotes | binding |
T315 | 1794-1801 | SO:0001091 | denotes | binding |
T316 | 1794-1801 | GO:0005488 | denotes | binding |
T340 | 1812-1815 | CHEBI:52242 | denotes | PTP |
T354 | 1812-1817 | P20417 | denotes | PTP1B |
T355 | 1812-1817 | P35821 | denotes | PTP1B |
T356 | 1812-1817 | PR:O13016 | denotes | PTP1B |
T357 | 1812-1817 | P18031 | denotes | PTP1B |
T358 | 1812-1817 | O13016 | denotes | PTP1B |
T359 | 1812-1817 | PR:000013448 | denotes | PTP1B |
T360 | 1812-1817 | PR:P18031 | denotes | PTP1B |
T361 | 1824-1835 | D005959 | denotes | glucosidase |
T362 | 1903-1910 | SO:0100018 | denotes | binding |
T363 | 1903-1910 | SO:0001091 | denotes | binding |
T364 | 1903-1910 | GO:0005488 | denotes | binding |
T365 | 2074-2090 | D000074385 | denotes | food ingredients |
T366 | 2074-2090 | D000074385 | denotes | food ingredients |
T367 | 2127-2142 | D003924 | denotes | type 2 diabetes |
T368 | 2127-2142 | D003924 | denotes | type 2 diabetes |
PubMed_ArguminSci
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 136-257 | DRI_Background | denotes | Sargassum serratifolium C. Agardh (Phaeophyceae, Fucales) is a marine brown alga that belongs to the family Sargassaceae. |
T2 | 258-327 | DRI_Background | denotes | It is widely distributed throughout coastal areas of Korea and Japan. |
T3 | 328-502 | DRI_Background | denotes | S. serratifolium has been found to contain high concentrations of plastoquinones, which have strong anti-cancer, anti-inflammatory, antioxidant, and neuroprotective activity. |
T4 | 503-723 | DRI_Background | denotes | This study aims to investigate the anti-diabetic activity of S. serratifolium and its major constituents through inhibition of protein tyrosine phosphatase 1B (PTP1B), α-glucosidase, and ONOO--mediated albumin nitration. |
T5 | 724-726 | DRI_Background | denotes | S. |
T6 | 751-853 | DRI_Background | denotes | extract and fractions exhibited broad PTP1B and α-glucosidase inhibitory activity (IC50, 1.83~7.04 and |
T7 | 871-914 | DRI_Background | denotes | for PTP1B and α-glucosidase, respectively). |
T8 | 915-1114 | DRI_Background | denotes | In an attempt to identify bioactive compounds, three plastoquinones (sargahydroquinoic acid, sargachromenol and sargaquinoic acid) were isolated from the active n-hexane fraction of S. serratifolium. |
T9 | 1115-1219 | DRI_Outcome | denotes | All three plastoquinones exhibited dose-dependent inhibitory activity against PTP1B in the IC50 range of |
T10 | 1233-1396 | DRI_Outcome | denotes | , while sargachromenol and sargaquinoic acid showed dose-dependent inhibitory activity against α-glucosidase (IC50 42.41 ± 3.09 and 96.17 ± 3.48 µM, respectively). |
T11 | 1397-1585 | DRI_Background | denotes | In the kinetic study of PTP1B enzyme inhibition, sargahydroquinoic acid and sargaquinoic acid led to mixed-type inhibition, whereas sargachromenol displayed noncompetitive-type inhibition. |
T12 | 1672-1959 | DRI_Approach | denotes | Docking simulations of these plastoquinones demonstrated negative binding energies and close proximity to residues in the binding pocket of PTP1B and α-glucosidase, indicating that these plastoquinones have high affinity and tight binding capacity towards the active site of the enzymes. |
T13 | 1960-2143 | DRI_Background | denotes | These results demonstrate that S. serratifolium and its major plastoquinones may have the potential as functional food ingredients for the prevention and treatment of type 2 diabetes. |
Goldhamster2_Cellosaurus
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 61-69 | CVCL_C410|Hybridoma|Mus musculus | denotes | Activity |
T2 | 160-161 | CVCL_S361|Finite_cell_line|Mus musculus | denotes | C |
T3 | 197-198 | CVCL_6479|Finite_cell_line|Mus musculus | denotes | a |
T4 | 345-348 | CVCL_6758|Undefined_cell_line_type|Cricetulus griseus | denotes | has |
T5 | 345-348 | CVCL_E689|Transformed_cell_line|Homo sapiens | denotes | has |
T6 | 433-439 | CVCL_E025|Induced_pluripotent_stem_cell|Homo sapiens | denotes | cancer |
T7 | 493-501 | CVCL_C410|Hybridoma|Mus musculus | denotes | activity |
T8 | 552-560 | CVCL_C410|Hybridoma|Mus musculus | denotes | activity |
T9 | 824-832 | CVCL_C410|Hybridoma|Mus musculus | denotes | activity |
T10 | 868-870 | CVCL_F566|Transformed_cell_line|Homo sapiens | denotes | mL |
T11 | 868-870 | CVCL_W799|Cancer_cell_line|Homo sapiens | denotes | mL |
T12 | 918-920 | CVCL_8754|Cancer_cell_line|Homo sapiens | denotes | an |
T13 | 918-920 | CVCL_H241|Cancer_cell_line|Homo sapiens | denotes | an |
T14 | 1069-1075 | CVCL_C410|Hybridoma|Mus musculus | denotes | active |
T15 | 1176-1184 | CVCL_C410|Hybridoma|Mus musculus | denotes | activity |
T16 | 1311-1319 | CVCL_C410|Hybridoma|Mus musculus | denotes | activity |
T17 | 1932-1938 | CVCL_C410|Hybridoma|Mus musculus | denotes | active |
T18 | 2037-2040 | CVCL_E773|Transformed_cell_line|Homo sapiens | denotes | may |