PubMed:23241745
Annnotations
PubTator4TogoVar
Id | Subject | Object | Predicate | Lexical cue | proteinmutation |
---|---|---|---|---|---|
23241745_0 | 589-595 | ProteinMutation | denotes | R1441G | rs33939927 |
23241745_1 | 599-605 | ProteinMutation | denotes | G2019S | rs34637584 |
c_corpus
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T7 | 0-3 | SO:0001444 | denotes | Ser |
T5 | 0-3 | Q62230 | denotes | Ser |
T6 | 0-3 | PR:000001931 | denotes | Ser |
T9 | 0-3 | PR:P18168 | denotes | Ser |
T1 | 0-3 | CHEBI:32838 | denotes | Ser |
T2 | 0-3 | CHEBI:32839 | denotes | Ser |
T4 | 0-3 | CHEBI:29999 | denotes | Ser |
T8 | 0-3 | CHEBI:17115 | denotes | Ser |
T3 | 0-3 | GO:0005790 | denotes | Ser |
T10 | 34-43 | CHEBI:47867 | denotes | indicator |
T11 | 47-52 | PR:Q5S006 | denotes | LRRK2 |
T12 | 47-52 | PR:000003033 | denotes | LRRK2 |
T13 | 47-52 | PR:Q5S007 | denotes | LRRK2 |
T14 | 53-68 | GO:0016301 | denotes | kinase activity |
T16 | 143-150 | 6308 | denotes | leucine |
T17 | 143-150 | SO:0001437 | denotes | leucine |
T15 | 143-150 | CHEBI:15603 | denotes | leucine |
T18 | 143-150 | D007930 | denotes | leucine |
T19 | 143-150 | CHEBI:25017 | denotes | leucine |
T20 | 143-150 | D007930 | denotes | leucine |
T21 | 156-162 | SO:0001068 | denotes | repeat |
T22 | 173-178 | PR:Q5S006 | denotes | LRRK2 |
T23 | 173-178 | PR:000003033 | denotes | LRRK2 |
T24 | 173-178 | PR:Q5S007 | denotes | LRRK2 |
T25 | 180-184 | SO:0000704 | denotes | gene |
T30 | 223-242 | D010300 | denotes | Parkinson's disease |
T31 | 223-242 | D010300 | denotes | Parkinson's disease |
T34 | 331-346 | GO:0016301 | denotes | kinase activity |
T35 | 359-364 | PR:Q5S006 | denotes | LRRK2 |
T36 | 359-364 | PR:000003033 | denotes | LRRK2 |
T37 | 359-364 | PR:Q5S007 | denotes | LRRK2 |
T38 | 417-422 | PR:Q5S006 | denotes | LRRK2 |
T39 | 417-422 | PR:000003033 | denotes | LRRK2 |
T40 | 417-422 | PR:Q5S007 | denotes | LRRK2 |
T41 | 423-438 | GO:0016301 | denotes | kinase activity |
T42 | 468-473 | PR:Q5S006 | denotes | LRRK2 |
T43 | 468-473 | PR:000003033 | denotes | LRRK2 |
T44 | 468-473 | PR:Q5S007 | denotes | LRRK2 |
T45 | 494-500 | CVCL_U693 | denotes | on Ser |
T50 | 497-500 | Q62230 | denotes | Ser |
T51 | 497-500 | PR:000001931 | denotes | Ser |
T54 | 497-500 | PR:P18168 | denotes | Ser |
T48 | 497-500 | GO:0005790 | denotes | Ser |
T46 | 497-500 | CHEBI:32838 | denotes | Ser |
T47 | 497-500 | CHEBI:32839 | denotes | Ser |
T49 | 497-500 | CHEBI:29999 | denotes | Ser |
T53 | 497-500 | CHEBI:17115 | denotes | Ser |
T52 | 497-500 | SO:0001444 | denotes | Ser |
T55 | 594-600 | CHEBI:86642 | denotes | G/C, G |
T60 | 673-676 | Q62230 | denotes | Ser |
T61 | 673-676 | PR:000001931 | denotes | Ser |
T64 | 673-676 | PR:P18168 | denotes | Ser |
T58 | 673-676 | GO:0005790 | denotes | Ser |
T62 | 673-676 | SO:0001444 | denotes | Ser |
T56 | 673-676 | CHEBI:32838 | denotes | Ser |
T57 | 673-676 | CHEBI:32839 | denotes | Ser |
T59 | 673-676 | CHEBI:29999 | denotes | Ser |
T63 | 673-676 | CHEBI:17115 | denotes | Ser |
T65 | 704-712 | SO:0000109 | denotes | Mutation |
T72 | 716-719 | SO:0001444 | denotes | Ser |
T70 | 716-719 | Q62230 | denotes | Ser |
T71 | 716-719 | PR:000001931 | denotes | Ser |
T74 | 716-719 | PR:P18168 | denotes | Ser |
T66 | 716-719 | CHEBI:32838 | denotes | Ser |
T67 | 716-719 | CHEBI:32839 | denotes | Ser |
T69 | 716-719 | CHEBI:29999 | denotes | Ser |
T73 | 716-719 | CHEBI:17115 | denotes | Ser |
T68 | 716-719 | GO:0005790 | denotes | Ser |
T79 | 729-736 | 426 | denotes | alanine |
T80 | 729-736 | SO:0001435 | denotes | alanine |
T75 | 729-736 | D000409 | denotes | alanine |
T76 | 729-736 | D000409 | denotes | alanine |
T77 | 729-736 | CHEBI:16977 | denotes | alanine |
T78 | 729-736 | CHEBI:46217 | denotes | alanine |
T81 | 729-736 | CHEBI:16449 | denotes | alanine |
T82 | 773-778 | PR:Q5S006 | denotes | LRRK2 |
T83 | 773-778 | PR:000003033 | denotes | LRRK2 |
T84 | 773-778 | PR:Q5S007 | denotes | LRRK2 |
T85 | 795-802 | GO:0043005 | denotes | neurite |
T86 | 795-812 | GO:0031175 | denotes | neurite outgrowth |
T87 | 825-828 | 10116 | denotes | rat |
T91 | 825-828 | D051381 | denotes | rat |
T88 | 825-828 | PR:P63003-1 | denotes | rat |
T89 | 825-828 | PR:Q2G0B1 | denotes | rat |
T90 | 825-828 | PR:Q8VHJ4 | denotes | rat |
T92 | 829-838 | P02301 | denotes | embryonic |
T93 | 829-838 | PR:000029532 | denotes | embryonic |
T100 | 920-923 | SO:0001444 | denotes | Ser |
T98 | 920-923 | Q62230 | denotes | Ser |
T99 | 920-923 | PR:000001931 | denotes | Ser |
T102 | 920-923 | PR:P18168 | denotes | Ser |
T94 | 920-923 | CHEBI:32838 | denotes | Ser |
T95 | 920-923 | CHEBI:32839 | denotes | Ser |
T97 | 920-923 | CHEBI:29999 | denotes | Ser |
T101 | 920-923 | CHEBI:17115 | denotes | Ser |
T96 | 920-923 | GO:0005790 | denotes | Ser |
T103 | 961-966 | UBERON:6110636 | denotes | brain |
T104 | 961-966 | UBERON:0000955 | denotes | brain |
T105 | 979-984 | PR:Q5S006 | denotes | LRRK2 |
T106 | 979-984 | PR:000003033 | denotes | LRRK2 |
T107 | 979-984 | PR:Q5S007 | denotes | LRRK2 |
T108 | 985-1001 | GO:0033673 | denotes | kinase inhibitor |
T109 | 992-1001 | CHEBI:35222 | denotes | inhibitor |
T116 | 1014-1017 | SO:0001444 | denotes | Ser |
T114 | 1014-1017 | Q62230 | denotes | Ser |
T115 | 1014-1017 | PR:000001931 | denotes | Ser |
T118 | 1014-1017 | PR:P18168 | denotes | Ser |
T110 | 1014-1017 | CHEBI:32838 | denotes | Ser |
T111 | 1014-1017 | CHEBI:32839 | denotes | Ser |
T113 | 1014-1017 | CHEBI:29999 | denotes | Ser |
T117 | 1014-1017 | CHEBI:17115 | denotes | Ser |
T112 | 1014-1017 | GO:0005790 | denotes | Ser |
T119 | 1096-1101 | PR:Q5S006 | denotes | LRRK2 |
T120 | 1096-1101 | PR:000003033 | denotes | LRRK2 |
T121 | 1096-1101 | PR:Q5S007 | denotes | LRRK2 |
T126 | 1149-1152 | Q62230 | denotes | Ser |
T127 | 1149-1152 | PR:000001931 | denotes | Ser |
T130 | 1149-1152 | PR:P18168 | denotes | Ser |
T124 | 1149-1152 | GO:0005790 | denotes | Ser |
T128 | 1149-1152 | SO:0001444 | denotes | Ser |
T122 | 1149-1152 | CHEBI:32838 | denotes | Ser |
T123 | 1149-1152 | CHEBI:32839 | denotes | Ser |
T125 | 1149-1152 | CHEBI:29999 | denotes | Ser |
T129 | 1149-1152 | CHEBI:17115 | denotes | Ser |
T131 | 1195-1204 | CHEBI:47867 | denotes | indicator |
T132 | 1208-1213 | PR:Q5S006 | denotes | LRRK2 |
T133 | 1208-1213 | PR:000003033 | denotes | LRRK2 |
T134 | 1208-1213 | PR:Q5S007 | denotes | LRRK2 |
T135 | 1214-1229 | GO:0016301 | denotes | kinase activity |
Allie
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
SS1_23241745_1_0 | 143-171 | expanded | denotes | leucine-rich repeat kinase 2 |
SS2_23241745_1_0 | 173-178 | abbr | denotes | LRRK2 |
SS1_23241745_1_1 | 223-242 | expanded | denotes | Parkinson's disease |
SS2_23241745_1_1 | 244-246 | abbr | denotes | PD |
SS1_23241745_5_0 | 716-736 | expanded | denotes | Ser(1292) to alanine |
SS2_23241745_5_0 | 738-744 | abbr | denotes | S1292A |
AE1_23241745_1_0 | SS1_23241745_1_0 | SS2_23241745_1_0 | abbreviatedTo | leucine-rich repeat kinase 2,LRRK2 |
AE1_23241745_1_1 | SS1_23241745_1_1 | SS2_23241745_1_1 | abbreviatedTo | Parkinson's disease,PD |
AE1_23241745_5_0 | SS1_23241745_5_0 | SS2_23241745_5_0 | abbreviatedTo | Ser(1292) to alanine,S1292A |
UseCases_ArguminSci_Discourse
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 0-125 | DRI_Background | denotes | Ser1292 autophosphorylation is an indicator of LRRK2 kinase activity and contributes to the cellular effects of PD mutations. |
T2 | 126-248 | DRI_Approach | denotes | Mutations in the leucine-rich repeat kinase 2 (LRRK2) gene are the most common cause of familial Parkinson's disease (PD). |
T3 | 249-447 | DRI_Background | denotes | Although biochemical studies have shown that certain PD mutations confer elevated kinase activity in vitro on LRRK2, there are no methods available to directly monitor LRRK2 kinase activity in vivo. |
T4 | 448-618 | DRI_Outcome | denotes | We demonstrate that LRRK2 autophosphorylation on Ser(1292) occurs in vivo and is enhanced by several familial PD mutations including N1437H, R1441G/C, G2019S, and I2020T. |
T5 | 619-703 | DRI_Approach | denotes | Combining two PD mutations together further increases Ser(1292) autophosphorylation. |
T6 | 704-855 | DRI_Background | denotes | Mutation of Ser(1292) to alanine (S1292A) ameliorates the effects of LRRK2 PD mutations on neurite outgrowth in cultured rat embryonic primary neurons. |
T7 | 856-960 | DRI_Outcome | denotes | Using cell-based and pharmacodynamic assays with phosphorylated Ser(1292) as the readout, we developed a |
T8 | 961-984 | Token_Label.OUTSIDE | denotes | brain-penetrating LRRK2 |
T9 | 985-1124 | DRI_Outcome | denotes | kinase inhibitor that blocks Ser(1292) autophosphorylation in vivo and attenuates the cellular consequences of LRRK2 PD mutations in vitro. |
T10 | 1125-1305 | DRI_Outcome | denotes | These data suggest that Ser(1292) autophosphorylation may be a useful indicator of LRRK2 kinase activity in vivo and may contribute to the cellular effects of certain PD mutations. |
PubMed_ArguminSci
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 126-248 | DRI_Approach | denotes | Mutations in the leucine-rich repeat kinase 2 (LRRK2) gene are the most common cause of familial Parkinson's disease (PD). |
T2 | 249-447 | DRI_Background | denotes | Although biochemical studies have shown that certain PD mutations confer elevated kinase activity in vitro on LRRK2, there are no methods available to directly monitor LRRK2 kinase activity in vivo. |
T3 | 448-618 | DRI_Outcome | denotes | We demonstrate that LRRK2 autophosphorylation on Ser(1292) occurs in vivo and is enhanced by several familial PD mutations including N1437H, R1441G/C, G2019S, and I2020T. |
T4 | 619-703 | DRI_Approach | denotes | Combining two PD mutations together further increases Ser(1292) autophosphorylation. |
T5 | 704-855 | DRI_Background | denotes | Mutation of Ser(1292) to alanine (S1292A) ameliorates the effects of LRRK2 PD mutations on neurite outgrowth in cultured rat embryonic primary neurons. |
T6 | 856-960 | DRI_Outcome | denotes | Using cell-based and pharmacodynamic assays with phosphorylated Ser(1292) as the readout, we developed a |
T7 | 985-1124 | DRI_Outcome | denotes | kinase inhibitor that blocks Ser(1292) autophosphorylation in vivo and attenuates the cellular consequences of LRRK2 PD mutations in vitro. |
T8 | 1125-1305 | DRI_Outcome | denotes | These data suggest that Ser(1292) autophosphorylation may be a useful indicator of LRRK2 kinase activity in vivo and may contribute to the cellular effects of certain PD mutations. |
PubmedHPO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 223-232 | HP_0001300 | denotes | Parkinson |
DisGeNET5_gene_disease
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
23241745-7#83#88#gene120892 | 1208-1213 | gene120892 | denotes | LRRK2 |
23241745-7#167#169#diseaseC0030567 | 1292-1294 | diseaseC0030567 | denotes | PD |
83#88#gene120892167#169#diseaseC0030567 | 23241745-7#83#88#gene120892 | 23241745-7#167#169#diseaseC0030567 | associated_with | LRRK2,PD |