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PubMed:18593936 JSONTXT

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PMID_GLOBAL

Id Subject Object Predicate Lexical cue mondo_id
T1 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer 0004986|0022578
T3 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer 0004986|0022578
T5 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor 0004987
T6 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer 0004986|0022578

LitCoin-entities-OrganismTaxon-PD

Id Subject Object Predicate Lexical cue db_id
T1 930-933 OrganismTaxon denotes Sp4 NCBItxid:10855
T2 1038-1041 OrganismTaxon denotes Sp4 NCBItxid:10855
T3 1292-1296 OrganismTaxon denotes mice NCBItxid:10095|NCBItxid:10088
T5 1381-1384 OrganismTaxon denotes Sp4 NCBItxid:10855

LitCoin-sentences

Id Subject Object Predicate Lexical cue
T8 1411-1637 Sentence denotes These results show for the first time that one of the underlying mechanisms of action of curcumin as a cancer chemotherapeutic agent is due, in part, to decreased expression of Sp transcription factors in bladder cancer cells.
T1 0-74 Sentence denotes Curcumin decreases specificity protein expression in bladder cancer cells.
T2 75-250 Sentence denotes Curcumin is the active component of tumeric, and this polyphenolic compound has been extensively investigated as an anticancer drug that modulates multiple pathways and genes.
T3 251-561 Sentence denotes In this study, 10 to 25 micromol/L curcumin inhibited 253JB-V and KU7 bladder cancer cell growth, and this was accompanied by induction of apoptosis and decreased expression of the proapoptotic protein survivin and the angiogenic proteins vascular endothelial growth factor (VEGF) and VEGF receptor 1 (VEGFR1).
T4 562-836 Sentence denotes Because expression of survivin, VEGF, and VEGFR1 are dependent on specificity protein (Sp) transcription factors, we also investigated the effects of curcumin on Sp protein expression as an underlying mechanism for the apoptotic and antiangiogenic activity of this compound.
T5 837-959 Sentence denotes The results show that curcumin induced proteasome-dependent down-regulation of Sp1, Sp3, and Sp4 in 253JB-V and KU7 cells.
T6 960-1230 Sentence denotes Moreover, using RNA interference with small inhibitory RNAs for Sp1, Sp3, and Sp4, we observed that curcumin-dependent inhibition of nuclear factor kappaB (NF-kappaB)-dependent genes, such as bcl-2, survivin, and cyclin D1, was also due, in part, to loss of Sp proteins.
T7 1231-1410 Sentence denotes Curcumin also decreased bladder tumor growth in athymic nude mice bearing KU7 cells as xenografts and this was accompanied by decreased Sp1, Sp3, and Sp4 protein levels in tumors.

LitCoin-entities

Id Subject Object Predicate Lexical cue db_id
5277 0-8 ChemicalEntity denotes Curcumin MESH:D003474
5278 19-38 GeneOrGeneProduct denotes specificity protein NCBIGene:6667|NCBIGene:6670|NCBIGene:6671
5279 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer MESH:D001749
5280 75-83 ChemicalEntity denotes Curcumin MESH:D003474
5281 286-294 ChemicalEntity denotes curcumin MESH:D003474
5282 305-312 CellLine denotes 253JB-V NCBITaxon:9606
5283 317-320 CellLine denotes KU7 NCBITaxon:9606
5284 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer MESH:D001749
5285 432-452 GeneOrGeneProduct denotes proapoptotic protein NCBIGene:332
5286 453-461 GeneOrGeneProduct denotes survivin NCBIGene:332
5287 470-489 GeneOrGeneProduct denotes angiogenic proteins NCBIGene:2321|NCBIGene:7422
5288 490-524 GeneOrGeneProduct denotes vascular endothelial growth factor NCBIGene:7422
5289 526-530 GeneOrGeneProduct denotes VEGF NCBIGene:7422
5290 536-551 GeneOrGeneProduct denotes VEGF receptor 1 NCBIGene:2321
5291 553-559 GeneOrGeneProduct denotes VEGFR1 NCBIGene:2321
5292 584-592 GeneOrGeneProduct denotes survivin NCBIGene:332
5293 594-598 GeneOrGeneProduct denotes VEGF NCBIGene:7422
5294 604-610 GeneOrGeneProduct denotes VEGFR1 NCBIGene:2321
5295 628-674 GeneOrGeneProduct denotes specificity protein (Sp) transcription factors NCBIGene:6667|NCBIGene:6670|NCBIGene:6671
5296 712-720 ChemicalEntity denotes curcumin MESH:D003474
5297 724-726 GeneOrGeneProduct denotes Sp NCBIGene:6667|NCBIGene:6670|NCBIGene:6671
5298 859-867 ChemicalEntity denotes curcumin MESH:D003474
5299 876-886 GeneOrGeneProduct denotes proteasome NCBIGene:5698
5300 916-919 GeneOrGeneProduct denotes Sp1 NCBIGene:6667
5301 921-924 GeneOrGeneProduct denotes Sp3 NCBIGene:6670
5302 930-933 GeneOrGeneProduct denotes Sp4 NCBIGene:6671
5303 937-944 CellLine denotes 253JB-V NCBITaxon:9606
5304 949-952 CellLine denotes KU7 NCBITaxon:9606
5305 1024-1027 GeneOrGeneProduct denotes Sp1 NCBIGene:6667
5306 1029-1032 GeneOrGeneProduct denotes Sp3 NCBIGene:6670
5307 1038-1041 GeneOrGeneProduct denotes Sp4 NCBIGene:6671
5308 1060-1068 ChemicalEntity denotes curcumin MESH:D003474
5309 1093-1114 GeneOrGeneProduct denotes nuclear factor kappaB NCBIGene:4790
5310 1116-1125 GeneOrGeneProduct denotes NF-kappaB NCBIGene:4790
5311 1152-1157 GeneOrGeneProduct denotes bcl-2 NCBIGene:596
5312 1159-1167 GeneOrGeneProduct denotes survivin NCBIGene:332
5313 1173-1182 GeneOrGeneProduct denotes cyclin D1 NCBIGene:595
5314 1218-1220 GeneOrGeneProduct denotes Sp NCBIGene:6667|NCBIGene:6670|NCBIGene:6671
5315 1231-1239 ChemicalEntity denotes Curcumin MESH:D003474
5316 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor MESH:D001749
5317 1292-1296 OrganismTaxon denotes mice NCBITaxon:10090
5318 1305-1308 CellLine denotes KU7 NCBITaxon:9606
5319 1367-1370 GeneOrGeneProduct denotes Sp1 NCBIGene:20683
5320 1372-1375 GeneOrGeneProduct denotes Sp3 NCBIGene:20687
5321 1381-1384 GeneOrGeneProduct denotes Sp4 NCBIGene:20688
5322 1403-1409 DiseaseOrPhenotypicFeature denotes tumors MESH:D009369
5323 1500-1508 ChemicalEntity denotes curcumin MESH:D003474
5324 1514-1520 DiseaseOrPhenotypicFeature denotes cancer MESH:D009369
5325 1588-1612 GeneOrGeneProduct denotes Sp transcription factors NCBIGene:6667|NCBIGene:6670|NCBIGene:6671
5326 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer MESH:D001749

LitCoin_Mondo

Id Subject Object Predicate Lexical cue mondo_id
T1 61-67 DiseaseOrPhenotypicFeature denotes cancer 0004992
T2 329-335 DiseaseOrPhenotypicFeature denotes cancer 0004992
T3 499-510 DiseaseOrPhenotypicFeature denotes endothelial 0015292
T4 1514-1520 DiseaseOrPhenotypicFeature denotes cancer 0004992
T5 1624-1630 DiseaseOrPhenotypicFeature denotes cancer 0004992

LitCoin-SeqVar

Id Subject Object Predicate Lexical cue
T1 305-310 SequenceVariant denotes 253JB
T2 937-942 SequenceVariant denotes 253JB

LitCoin-GeneOrGeneProduct-v0

Id Subject Object Predicate Lexical cue
T1 31-38 GeneOrGeneProduct denotes protein
T2 68-73 GeneOrGeneProduct denotes cells
T3 91-97 GeneOrGeneProduct denotes active
T4 160-171 GeneOrGeneProduct denotes extensively
T5 222-230 GeneOrGeneProduct denotes multiple
T6 336-340 GeneOrGeneProduct denotes cell
T7 341-347 GeneOrGeneProduct denotes growth
T8 390-399 GeneOrGeneProduct denotes apoptosis
T9 445-452 GeneOrGeneProduct denotes protein
T10 453-461 GeneOrGeneProduct denotes survivin
T11 481-489 GeneOrGeneProduct denotes proteins
T12 490-524 GeneOrGeneProduct denotes vascular endothelial growth factor
T13 526-530 GeneOrGeneProduct denotes VEGF
T14 536-549 GeneOrGeneProduct denotes VEGF receptor
T15 553-559 GeneOrGeneProduct denotes VEGFR1
T16 584-592 GeneOrGeneProduct denotes survivin
T17 594-598 GeneOrGeneProduct denotes VEGF
T18 604-610 GeneOrGeneProduct denotes VEGFR1
T19 640-647 GeneOrGeneProduct denotes protein
T20 653-674 GeneOrGeneProduct denotes transcription factors
T21 727-734 GeneOrGeneProduct denotes protein
T22 810-818 GeneOrGeneProduct denotes activity
T23 868-875 GeneOrGeneProduct denotes induced
T24 876-886 GeneOrGeneProduct denotes proteasome
T25 902-912 GeneOrGeneProduct denotes regulation
T26 916-919 GeneOrGeneProduct denotes Sp1
T27 921-924 GeneOrGeneProduct denotes Sp3
T28 930-933 GeneOrGeneProduct denotes Sp4
T29 953-958 GeneOrGeneProduct denotes cells
T30 998-1003 GeneOrGeneProduct denotes small
T31 1024-1027 GeneOrGeneProduct denotes Sp1
T32 1029-1032 GeneOrGeneProduct denotes Sp3
T33 1038-1041 GeneOrGeneProduct denotes Sp4
T34 1101-1107 GeneOrGeneProduct denotes factor
T35 1116-1125 GeneOrGeneProduct denotes NF-kappaB
T36 1152-1157 GeneOrGeneProduct denotes bcl-2
T37 1159-1167 GeneOrGeneProduct denotes survivin
T38 1173-1182 GeneOrGeneProduct denotes cyclin D1
T39 1201-1205 GeneOrGeneProduct denotes part
T40 1221-1229 GeneOrGeneProduct denotes proteins
T41 1263-1268 GeneOrGeneProduct denotes tumor
T42 1269-1275 GeneOrGeneProduct denotes growth
T43 1287-1291 GeneOrGeneProduct denotes nude
T44 1292-1296 GeneOrGeneProduct denotes mice
T45 1309-1314 GeneOrGeneProduct denotes cells
T46 1367-1370 GeneOrGeneProduct denotes Sp1
T47 1372-1375 GeneOrGeneProduct denotes Sp3
T48 1385-1392 GeneOrGeneProduct denotes protein
T49 1403-1409 GeneOrGeneProduct denotes tumors
T50 1444-1448 GeneOrGeneProduct denotes time
T51 1555-1559 GeneOrGeneProduct denotes part
T52 1591-1612 GeneOrGeneProduct denotes transcription factors
T53 1631-1636 GeneOrGeneProduct denotes cells

LitCoin-GeneOrGeneProduct-v2

Id Subject Object Predicate Lexical cue
T1 31-38 GeneOrGeneProduct denotes protein
T2 222-230 GeneOrGeneProduct denotes multiple
T3 336-340 GeneOrGeneProduct denotes cell
T4 341-347 GeneOrGeneProduct denotes growth
T5 390-399 GeneOrGeneProduct denotes apoptosis
T6 445-452 GeneOrGeneProduct denotes protein
T7 453-461 GeneOrGeneProduct denotes survivin
T8 490-524 GeneOrGeneProduct denotes vascular endothelial growth factor
T9 526-530 GeneOrGeneProduct denotes VEGF
T10 536-549 GeneOrGeneProduct denotes VEGF receptor
T11 553-559 GeneOrGeneProduct denotes VEGFR1
T12 584-592 GeneOrGeneProduct denotes survivin
T13 594-598 GeneOrGeneProduct denotes VEGF
T14 604-610 GeneOrGeneProduct denotes VEGFR1
T15 640-647 GeneOrGeneProduct denotes protein
T16 653-674 GeneOrGeneProduct denotes transcription factors
T17 727-734 GeneOrGeneProduct denotes protein
T18 876-886 GeneOrGeneProduct denotes proteasome
T19 998-1003 GeneOrGeneProduct denotes small
T20 1101-1107 GeneOrGeneProduct denotes factor
T21 1116-1125 GeneOrGeneProduct denotes NF-kappaB
T22 1152-1157 GeneOrGeneProduct denotes bcl-2
T23 1159-1167 GeneOrGeneProduct denotes survivin
T24 1173-1182 GeneOrGeneProduct denotes cyclin D1
T25 1269-1275 GeneOrGeneProduct denotes growth
T26 1287-1291 GeneOrGeneProduct denotes nude
T27 1385-1392 GeneOrGeneProduct denotes protein
T28 1591-1612 GeneOrGeneProduct denotes transcription factors

LitCoin-Disease-MeSH

Id Subject Object Predicate Lexical cue originalLabel
T1 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T2 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T3 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor D001749
T4 1403-1409 DiseaseOrPhenotypicFeature denotes tumors D009369
T5 1514-1520 DiseaseOrPhenotypicFeature denotes cancer D009369
T6 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer D001749

LitCoin_Mondo_095

Id Subject Object Predicate Lexical cue mondo_id
T1 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer 0022578|0004986
T3 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer 0022578|0004986
T5 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor 0004987
T6 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer 0022578|0004986

LitCoin-MeSH-Disease-2

Id Subject Object Predicate Lexical cue ID:
T1 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T2 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T3 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor D001749
T4 1403-1409 DiseaseOrPhenotypicFeature denotes tumors DISEASE|D009369
T6 1514-1520 DiseaseOrPhenotypicFeature denotes cancer D009369
T7 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer D001749

LitCoin_CellLine

Id Subject Object Predicate Lexical cue cellosaurus_accession_id
T1 305-312 CellLine denotes 253JB-V CVCL_7937
T2 317-320 CellLine denotes KU7 CVCL_4714|CVCL_T528
T4 937-944 CellLine denotes 253JB-V CVCL_7937
T5 949-952 CellLine denotes KU7 CVCL_4714|CVCL_T528
T7 1305-1308 CellLine denotes KU7 CVCL_4714|CVCL_T528

LitCoin-MONDO_bioort2019

Id Subject Object Predicate Lexical cue #label
T1 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T2 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T3 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor D001749
T4 1403-1409 DiseaseOrPhenotypicFeature denotes tumors D009369
T5 1514-1520 DiseaseOrPhenotypicFeature denotes cancer D009369
T6 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer D001749

LitCoin-Chemical-MeSH-CHEBI

Id Subject Object Predicate Lexical cue ID:
T1 0-8 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T2 75-83 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T3 286-294 ChemicalEntity denotes curcumin D003474|http://purl.obolibrary.org/obo/CHEBI_3962
T5 712-720 ChemicalEntity denotes curcumin D003474|http://purl.obolibrary.org/obo/CHEBI_3962
T7 859-867 ChemicalEntity denotes curcumin D003474|http://purl.obolibrary.org/obo/CHEBI_3962
T9 876-886 ChemicalEntity denotes proteasome D046988
T10 1060-1068 ChemicalEntity denotes curcumin D003474|http://purl.obolibrary.org/obo/CHEBI_3962
T12 1231-1239 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T13 1500-1508 ChemicalEntity denotes curcumin D003474|http://purl.obolibrary.org/obo/CHEBI_3962

LitCoin-NCBITaxon-2

Id Subject Object Predicate Lexical cue
T1 930-933 OrganismTaxon denotes Sp4
T2 1038-1041 OrganismTaxon denotes Sp4
T3 1292-1296 OrganismTaxon denotes mice
T4 1381-1384 OrganismTaxon denotes Sp4

LitCoin-GeneOrGeneProduct-v3

Id Subject Object Predicate Lexical cue
T1 31-52 GeneOrGeneProduct denotes protein expression in
T2 453-461 GeneOrGeneProduct denotes survivin
T3 490-524 GeneOrGeneProduct denotes vascular endothelial growth factor
T4 526-530 GeneOrGeneProduct denotes VEGF
T5 536-549 GeneOrGeneProduct denotes VEGF receptor
T7 553-559 GeneOrGeneProduct denotes VEGFR1
T8 584-592 GeneOrGeneProduct denotes survivin
T9 594-598 GeneOrGeneProduct denotes VEGF
T10 604-610 GeneOrGeneProduct denotes VEGFR1
T11 648-674 GeneOrGeneProduct denotes (Sp) transcription factors
T12 727-745 GeneOrGeneProduct denotes protein expression
T13 876-886 GeneOrGeneProduct denotes proteasome
T14 1093-1114 GeneOrGeneProduct denotes nuclear factor kappaB
T15 1116-1125 GeneOrGeneProduct denotes NF-kappaB
T16 1152-1157 GeneOrGeneProduct denotes bcl-2
T17 1159-1167 GeneOrGeneProduct denotes survivin
T18 1173-1182 GeneOrGeneProduct denotes cyclin D1
T19 1381-1392 GeneOrGeneProduct denotes Sp4 protein
T20 1588-1612 GeneOrGeneProduct denotes Sp transcription factors

LitCoin-training-merged

Id Subject Object Predicate Lexical cue #label ID: cellosaurus_accession_id
T7 1305-1308 CellLine denotes KU7 CVCL_T528|CVCL_4714
T5 949-952 CellLine denotes KU7 CVCL_T528|CVCL_4714
T4 937-944 CellLine denotes 253JB-V CVCL_7937
T2 317-320 CellLine denotes KU7 CVCL_T528|CVCL_4714
T1 305-312 CellLine denotes 253JB-V CVCL_7937
T13 1500-1508 ChemicalEntity denotes curcumin http://purl.obolibrary.org/obo/CHEBI_3962|D003474
T12 1231-1239 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T10 1060-1068 ChemicalEntity denotes curcumin http://purl.obolibrary.org/obo/CHEBI_3962|D003474
T9 876-886 ChemicalEntity denotes proteasome D046988
T73698 859-867 ChemicalEntity denotes curcumin http://purl.obolibrary.org/obo/CHEBI_3962|D003474
T20223 712-720 ChemicalEntity denotes curcumin http://purl.obolibrary.org/obo/CHEBI_3962|D003474
T3 286-294 ChemicalEntity denotes curcumin http://purl.obolibrary.org/obo/CHEBI_3962|D003474
T53129 75-83 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T58180 0-8 ChemicalEntity denotes Curcumin http://purl.obolibrary.org/obo/CHEBI_3962
T20 1588-1612 GeneOrGeneProduct denotes Sp transcription factors
T19 1381-1392 GeneOrGeneProduct denotes Sp4 protein
T18 1173-1182 GeneOrGeneProduct denotes cyclin D1
T17 1159-1167 GeneOrGeneProduct denotes survivin
T16 1152-1157 GeneOrGeneProduct denotes bcl-2
T15 1116-1125 GeneOrGeneProduct denotes NF-kappaB
T14 1093-1114 GeneOrGeneProduct denotes nuclear factor kappaB
T90268 876-886 GeneOrGeneProduct denotes proteasome
T57130 727-745 GeneOrGeneProduct denotes protein expression
T11 648-674 GeneOrGeneProduct denotes (Sp) transcription factors
T62110 604-610 GeneOrGeneProduct denotes VEGFR1
T99500 594-598 GeneOrGeneProduct denotes VEGF
T8 584-592 GeneOrGeneProduct denotes survivin
T25680 553-559 GeneOrGeneProduct denotes VEGFR1
T16794 536-549 GeneOrGeneProduct denotes VEGF receptor
T51465 526-530 GeneOrGeneProduct denotes VEGF
T40850 490-524 GeneOrGeneProduct denotes vascular endothelial growth factor
T85350 453-461 GeneOrGeneProduct denotes survivin
T25491 31-52 GeneOrGeneProduct denotes protein expression in
T6 1616-1630 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T92657 1514-1520 DiseaseOrPhenotypicFeature denotes cancer D009369
T69113 1403-1409 DiseaseOrPhenotypicFeature denotes tumors D009369
T73033 1255-1268 DiseaseOrPhenotypicFeature denotes bladder tumor D001749
T12719 321-335 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T45542 53-67 DiseaseOrPhenotypicFeature denotes bladder cancer D001749
T94703 1381-1384 OrganismTaxon denotes Sp4
T14117 1292-1296 OrganismTaxon denotes mice
T20516 1038-1041 OrganismTaxon denotes Sp4
T11231 930-933 OrganismTaxon denotes Sp4
T34723 937-942 SequenceVariant denotes 253JB
T87809 305-310 SequenceVariant denotes 253JB

DisGeNET

Id Subject Object Predicate Lexical cue
T0 1381-1384 gene:6671 denotes Sp4
T1 1255-1268 disease:C0005695 denotes bladder tumor
R1 T0 T1 associated_with Sp4,bladder tumor

DisGeNET5_gene_disease

Id Subject Object Predicate Lexical cue
18593936-6#150#153#gene6671 1381-1384 gene6671 denotes Sp4
18593936-6#24#37#diseaseC0005695 1255-1268 diseaseC0005695 denotes bladder tumor
150#153#gene667124#37#diseaseC0005695 18593936-6#150#153#gene6671 18593936-6#24#37#diseaseC0005695 associated_with Sp4,bladder tumor