PubMed:1310680
Annnotations
sentences
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-75 | Sentence | denotes | Structure function analysis of vitamin D analogs with C-ring modifications. |
| T2 | 76-183 | Sentence | denotes | Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3) with substitutions on C-11 were synthesized. |
| T3 | 184-532 | Sentence | denotes | Small apolar substitutions (11 alpha-methyl, 11 alpha-fluoromethyl) did not markedly decrease the affinity for the vitamin D receptor, but larger (11 alpha-chloromethyl or 11 alpha- or 11 beta-phenyl) or more polar substitutions (11 alpha-hydroxymethyl, 11 alpha-(2-hydroxyethyl] decreased the affinity to less than 5% of that of 1 alpha,25-OH)2D3. |
| T4 | 533-615 | Sentence | denotes | Their affinity for the vitamin D-binding protein, however, increased up to 4-fold. |
| T5 | 616-902 | Sentence | denotes | The biological activity of 11 alpha-methyl-1 alpha,25-(OH)2D3 closely resembled that of the natural hormone on normal and leukemic cell proliferation and bone resorption, whereas its in vivo effect on calcium metabolism of the rachitic chick was about 50% of that of 1 alpha,25-(OH)2D3. |
| T6 | 903-971 | Sentence | denotes | The 11 beta-methyl analog had a greater than 10-fold lower activity. |
| T7 | 972-1192 | Sentence | denotes | The differentiating effects of the other C-11 analogs on human promyeloid leukemia cells (HL-60) agreed well with their bone-resorbing activity and receptor affinity, but they demonstrated lower calcemic effects in vivo. |
| T8 | 1193-1357 | Sentence | denotes | Large or polar substitutions on C-11 of 1 alpha,25-(OH)2D3 thus impair the binding of the vitamin D receptor but increase the affinity to vitamin D-binding protein. |
| T9 | 1358-1498 | Sentence | denotes | The effects of many C-11-substituted 1 alpha,25-(OH)2D3 analogs on HL-60 cell differentiation exceeded their activity on calcium metabolism. |
| T1 | 0-75 | Sentence | denotes | Structure function analysis of vitamin D analogs with C-ring modifications. |
| T2 | 76-183 | Sentence | denotes | Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3) with substitutions on C-11 were synthesized. |
| T3 | 184-532 | Sentence | denotes | Small apolar substitutions (11 alpha-methyl, 11 alpha-fluoromethyl) did not markedly decrease the affinity for the vitamin D receptor, but larger (11 alpha-chloromethyl or 11 alpha- or 11 beta-phenyl) or more polar substitutions (11 alpha-hydroxymethyl, 11 alpha-(2-hydroxyethyl] decreased the affinity to less than 5% of that of 1 alpha,25-OH)2D3. |
| T4 | 533-615 | Sentence | denotes | Their affinity for the vitamin D-binding protein, however, increased up to 4-fold. |
| T5 | 616-902 | Sentence | denotes | The biological activity of 11 alpha-methyl-1 alpha,25-(OH)2D3 closely resembled that of the natural hormone on normal and leukemic cell proliferation and bone resorption, whereas its in vivo effect on calcium metabolism of the rachitic chick was about 50% of that of 1 alpha,25-(OH)2D3. |
| T6 | 903-971 | Sentence | denotes | The 11 beta-methyl analog had a greater than 10-fold lower activity. |
| T7 | 972-1192 | Sentence | denotes | The differentiating effects of the other C-11 analogs on human promyeloid leukemia cells (HL-60) agreed well with their bone-resorbing activity and receptor affinity, but they demonstrated lower calcemic effects in vivo. |
| T8 | 1193-1357 | Sentence | denotes | Large or polar substitutions on C-11 of 1 alpha,25-(OH)2D3 thus impair the binding of the vitamin D receptor but increase the affinity to vitamin D-binding protein. |
| T9 | 1358-1498 | Sentence | denotes | The effects of many C-11-substituted 1 alpha,25-(OH)2D3 analogs on HL-60 cell differentiation exceeded their activity on calcium metabolism. |
Glycosmos6-MAT
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 770-774 | http://purl.obolibrary.org/obo/MAT_0000299 | denotes | bone |
| T2 | 1092-1096 | http://purl.obolibrary.org/obo/MAT_0000299 | denotes | bone |
jnlpba-st-training
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 299-317 | protein | denotes | vitamin D receptor |
| T2 | 556-581 | protein | denotes | vitamin D-binding protein |
| T3 | 738-751 | cell_type | denotes | leukemic cell |
| T4 | 1029-1060 | cell_line | denotes | human promyeloid leukemia cells |
| T5 | 1062-1067 | cell_line | denotes | HL-60 |
| T6 | 1283-1301 | protein | denotes | vitamin D receptor |
| T7 | 1331-1356 | protein | denotes | vitamin D-binding protein |
| T8 | 1425-1430 | cell_line | denotes | HL-60 |
pubmed-sentences-benchmark
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| S1 | 0-75 | Sentence | denotes | Structure function analysis of vitamin D analogs with C-ring modifications. |
| S2 | 76-183 | Sentence | denotes | Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3) with substitutions on C-11 were synthesized. |
| S3 | 184-532 | Sentence | denotes | Small apolar substitutions (11 alpha-methyl, 11 alpha-fluoromethyl) did not markedly decrease the affinity for the vitamin D receptor, but larger (11 alpha-chloromethyl or 11 alpha- or 11 beta-phenyl) or more polar substitutions (11 alpha-hydroxymethyl, 11 alpha-(2-hydroxyethyl] decreased the affinity to less than 5% of that of 1 alpha,25-OH)2D3. |
| S4 | 533-615 | Sentence | denotes | Their affinity for the vitamin D-binding protein, however, increased up to 4-fold. |
| S5 | 616-902 | Sentence | denotes | The biological activity of 11 alpha-methyl-1 alpha,25-(OH)2D3 closely resembled that of the natural hormone on normal and leukemic cell proliferation and bone resorption, whereas its in vivo effect on calcium metabolism of the rachitic chick was about 50% of that of 1 alpha,25-(OH)2D3. |
| S6 | 903-971 | Sentence | denotes | The 11 beta-methyl analog had a greater than 10-fold lower activity. |
| S7 | 972-1192 | Sentence | denotes | The differentiating effects of the other C-11 analogs on human promyeloid leukemia cells (HL-60) agreed well with their bone-resorbing activity and receptor affinity, but they demonstrated lower calcemic effects in vivo. |
| S8 | 1193-1357 | Sentence | denotes | Large or polar substitutions on C-11 of 1 alpha,25-(OH)2D3 thus impair the binding of the vitamin D receptor but increase the affinity to vitamin D-binding protein. |
| S9 | 1358-1498 | Sentence | denotes | The effects of many C-11-substituted 1 alpha,25-(OH)2D3 analogs on HL-60 cell differentiation exceeded their activity on calcium metabolism. |
genia-medco-coref
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| C1 | 31-48 | NP | denotes | vitamin D analogs |
| C3 | 87-138 | NP | denotes | 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3) |
| C2 | 76-138 | NP | denotes | Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3) |
| C4 | 161-165 | NP | denotes | C-11 |
| C5 | 184-251 | NP | denotes | Small apolar substitutions (11 alpha-methyl, 11 alpha-fluoromethyl) |
| C7 | 295-317 | NP | denotes | the vitamin D receptor |
| C6 | 278-317 | NP | denotes | the affinity for the vitamin D receptor |
| C8 | 474-486 | NP | denotes | the affinity |
| C9 | 506-510 | NP | denotes | that |
| C10 | 514-531 | NP | denotes | 1 alpha,25-OH)2D3 |
| C11 | 533-538 | NP | denotes | Their |
| C12 | 552-581 | NP | denotes | the vitamin D-binding protein |
| C13 | 616-639 | NP | denotes | The biological activity |
| C14 | 643-677 | NP | denotes | 11 alpha-methyl-1 alpha,25-(OH)2D3 |
| C15 | 696-700 | NP | denotes | that |
| C16 | 795-798 | NP | denotes | its |
| C17 | 807-813 | NP | denotes | effect |
| C18 | 817-835 | NP | denotes | calcium metabolism |
| C19 | 875-879 | NP | denotes | that |
| C20 | 883-901 | NP | denotes | 1 alpha,25-(OH)2D3 |
| C22 | 1013-1017 | NP | denotes | C-11 |
| C21 | 1003-1025 | NP | denotes | the other C-11 analogs |
| C23 | 1086-1091 | NP | denotes | their |
| C24 | 1143-1147 | NP | denotes | they |
| C25 | 1225-1229 | NP | denotes | C-11 |
| C26 | 1233-1251 | NP | denotes | 1 alpha,25-(OH)2D3 |
| C27 | 1279-1301 | NP | denotes | the vitamin D receptor |
| C28 | 1331-1356 | NP | denotes | vitamin D-binding protein |
| C30 | 1395-1413 | NP | denotes | 1 alpha,25-(OH)2D3 |
| C29 | 1378-1421 | NP | denotes | C-11-substituted 1 alpha,25-(OH)2D3 analogs |
| C31 | 1461-1466 | NP | denotes | their |
| C32 | 1479-1497 | NP | denotes | calcium metabolism |
| R1 | C2 | C1 | coref-ident | "Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3)",vitamin D analogs |
| R2 | C8 | C6 | coref-ident | the affinity,the affinity for the vitamin D receptor |
| R3 | C9 | C8 | coref-pron | that,the affinity |
| R4 | C10 | C3 | coref-ident | "1 alpha,25-OH)2D3","1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3)" |
| R5 | C11 | C5 | coref-pron | Their,"Small apolar substitutions (11 alpha-methyl, 11 alpha-fluoromethyl)" |
| R6 | C15 | C13 | coref-pron | that,The biological activity |
| R7 | C16 | C14 | coref-pron | its,"11 alpha-methyl-1 alpha,25-(OH)2D3" |
| R8 | C19 | C17 | coref-pron | that,effect |
| R9 | C20 | C10 | coref-ident | "1 alpha,25-(OH)2D3","1 alpha,25-OH)2D3" |
| R10 | C22 | C4 | coref-ident | C-11,C-11 |
| R11 | C23 | C21 | coref-pron | their,the other C-11 analogs |
| R12 | C24 | C21 | coref-pron | they,the other C-11 analogs |
| R13 | C25 | C22 | coref-ident | C-11,C-11 |
| R14 | C26 | C20 | coref-ident | "1 alpha,25-(OH)2D3","1 alpha,25-(OH)2D3" |
| R15 | C27 | C7 | coref-ident | the vitamin D receptor,the vitamin D receptor |
| R16 | C28 | C12 | coref-ident | vitamin D-binding protein,the vitamin D-binding protein |
| R17 | C30 | C26 | coref-ident | "1 alpha,25-(OH)2D3","1 alpha,25-(OH)2D3" |
| R18 | C29 | C2 | coref-other | "C-11-substituted 1 alpha,25-(OH)2D3 analogs","Analogs of 1 alpha,25-dihydroxyvitamin D3 (1 alpha,25-(OH)2D3)" |
| R19 | C31 | C29 | coref-pron | their,"C-11-substituted 1 alpha,25-(OH)2D3 analogs" |
| R20 | C32 | C18 | coref-ident | calcium metabolism,calcium metabolism |
GENIAcorpus
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 31-40 | lipid | denotes | vitamin D |
| T2 | 54-74 | other_name | denotes | C-ring modifications |
| T3 | 87-117 | lipid | denotes | 1 alpha,25-dihydroxyvitamin D3 |
| T4 | 119-137 | lipid | denotes | 1 alpha,25-(OH)2D3 |
| T5 | 161-165 | other_name | denotes | C-11 |
| T6 | 184-210 | other_name | denotes | Small apolar substitutions |
| T7 | 212-250 | lipid | denotes | 11 alpha-methyl, 11 alpha-fluoromethyl |
| T8 | 299-308 | lipid | denotes | vitamin D |
| T9 | 331-383 | lipid | denotes | 11 alpha-chloromethyl or 11 alpha- or 11 beta-phenyl |
| T10 | 414-462 | lipid | denotes | 11 alpha-hydroxymethyl, 11 alpha-(2-hydroxyethyl |
| T11 | 514-531 | lipid | denotes | 1 alpha,25-OH)2D3 |
| T12 | 556-565 | lipid | denotes | vitamin D |
| T13 | 643-677 | lipid | denotes | 11 alpha-methyl-1 alpha,25-(OH)2D3 |
| T14 | 738-751 | cell_type | denotes | leukemic cell |
| T15 | 817-824 | atom | denotes | calcium |
| T16 | 883-901 | lipid | denotes | 1 alpha,25-(OH)2D3 |
| T17 | 907-928 | lipid | denotes | 11 beta-methyl analog |
| T18 | 1013-1025 | lipid | denotes | C-11 analogs |
| T19 | 1029-1060 | cell_line | denotes | human promyeloid leukemia cells |
| T20 | 1062-1067 | cell_line | denotes | HL-60 |
| T21 | 1202-1221 | other_name | denotes | polar substitutions |
| T22 | 1225-1229 | lipid | denotes | C-11 |
| T23 | 1233-1251 | lipid | denotes | 1 alpha,25-(OH)2D3 |
| T24 | 1283-1292 | lipid | denotes | vitamin D |
| T25 | 1331-1356 | protein_family_or_group | denotes | vitamin D-binding protein |
| T26 | 1378-1394 | lipid | denotes | C-11-substituted |
| T27 | 1395-1413 | lipid | denotes | 1 alpha,25-(OH)2D3 |
| T28 | 1425-1430 | cell_line | denotes | HL-60 |
| T29 | 1479-1486 | atom | denotes | calcium |
Anatomy-MAT
| Id | Subject | Object | Predicate | Lexical cue | mat_id |
|---|---|---|---|---|---|
| T1 | 770-774 | Body_part | denotes | bone | http://purl.obolibrary.org/obo/MAT_0000299 |
| T2 | 1092-1096 | Body_part | denotes | bone | http://purl.obolibrary.org/obo/MAT_0000299 |
HP-phenotype
| Id | Subject | Object | Predicate | Lexical cue | hp_id |
|---|---|---|---|---|---|
| T1 | 1046-1054 | Phenotype | denotes | leukemia | HP:0001909 |
mondo_disease
| Id | Subject | Object | Predicate | Lexical cue | mondo_id |
|---|---|---|---|---|---|
| T1 | 1046-1054 | Disease | denotes | leukemia | http://purl.obolibrary.org/obo/MONDO_0005059 |
NCBITAXON
| Id | Subject | Object | Predicate | Lexical cue | db_id |
|---|---|---|---|---|---|
| T1 | 1029-1034 | OrganismTaxon | denotes | human | 9606 |
Anatomy-UBERON
| Id | Subject | Object | Predicate | Lexical cue | uberon_id |
|---|---|---|---|---|---|
| T1 | 770-774 | Body_part | denotes | bone | http://purl.obolibrary.org/obo/UBERON_0001474|http://purl.obolibrary.org/obo/UBERON_0002481 |
| T3 | 1092-1096 | Body_part | denotes | bone | http://purl.obolibrary.org/obo/UBERON_0001474|http://purl.obolibrary.org/obo/UBERON_0002481 |