PubMed:12297502
Annnotations
sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 0-123 | Sentence | denotes | Inhibition of silencing and accelerated aging by nicotinamide, a putative negative regulator of yeast sir2 and human SIRT1. |
T2 | 124-298 | Sentence | denotes | The Saccharomyces cerevisiae Sir2 protein is an NAD(+)-dependent histone deacetylase that plays a critical role in transcriptional silencing, genome stability, and longevity. |
T3 | 299-407 | Sentence | denotes | A human homologue of Sir2, SIRT1, regulates the activity of the p53 tumor suppressor and inhibits apoptosis. |
T4 | 408-566 | Sentence | denotes | The Sir2 deacetylation reaction generates two products: O-acetyl-ADP-ribose and nicotinamide, a precursor of nicotinic acid and a form of niacin/vitamin B(3). |
T5 | 567-723 | Sentence | denotes | We show here that nicotinamide strongly inhibits yeast silencing, increases rDNA recombination, and shortens replicative life span to that of a sir2 mutant. |
T6 | 724-909 | Sentence | denotes | Nicotinamide abolishes silencing and leads to an eventual delocalization of Sir2 even in G(1)-arrested cells, demonstrating that silent heterochromatin requires continual Sir2 activity. |
T7 | 910-1022 | Sentence | denotes | We show that physiological concentrations of nicotinamide noncompetitively inhibit both Sir2 and SIRT1 in vitro. |
T8 | 1023-1184 | Sentence | denotes | The degree of inhibition by nicotinamide (IC(50) < 50 microm) is equal to or better than the most effective known synthetic inhibitors of this class of proteins. |
T9 | 1185-1336 | Sentence | denotes | We propose a model whereby nicotinamide inhibits deacetylation by binding to a conserved pocket adjacent to NAD(+), thereby blocking NAD(+) hydrolysis. |
T10 | 1337-1438 | Sentence | denotes | We discuss the possibility that nicotinamide is a physiologically relevant regulator of Sir2 enzymes. |
PubmedHPO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 367-372 | HP_0002664 | denotes | tumor |
FSU-PRGE
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 102-106 | protein | denotes | sir2 |
T2 | 117-122 | protein | denotes | SIRT1 |
T3 | 153-157 | protein | denotes | Sir2 |
T4 | 189-208 | protein | denotes | histone deacetylase |
T5 | 320-324 | protein | denotes | Sir2 |
T6 | 326-331 | protein | denotes | SIRT1 |
T7 | 363-383 | protein | denotes | p53 tumor suppressor |
T8 | 412-416 | protein | denotes | Sir2 |
T9 | 711-715 | protein | denotes | sir2 |
T10 | 800-804 | protein | denotes | Sir2 |
T11 | 895-899 | protein | denotes | Sir2 |
T12 | 998-1002 | protein | denotes | Sir2 |
T13 | 1007-1012 | protein | denotes | SIRT1 |
T14 | 1425-1429 | protein | denotes | Sir2 |
PIR-corpus2
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 102-106 | protein | denotes | sir2 |
T2 | 117-122 | protein | denotes | SIRT1 |
T3 | 153-165 | protein | denotes | Sir2 protein |
T4 | 172-196 | protein | denotes | NAD(+)-dependent histone |
T5 | 320-324 | protein | denotes | Sir2 |
T6 | 326-331 | protein | denotes | SIRT1 |
T7 | 363-383 | protein | denotes | p53 tumor suppressor |
T8 | 412-416 | protein | denotes | Sir2 |
T9 | 711-715 | protein | denotes | sir2 |
T10 | 800-804 | protein | denotes | Sir2 |
T11 | 895-899 | protein | denotes | Sir2 |
T12 | 998-1002 | protein | denotes | Sir2 |
T13 | 1007-1012 | protein | denotes | SIRT1 |
T14 | 1425-1437 | protein | denotes | Sir2 enzymes |
T19 | 111-122 | long_form | denotes | human SIRT1 |
PIR-corpus1
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T1 | 153-165 | protein | denotes | Sir2 protein |
T2 | 172-196 | protein | denotes | NAD(+)-dependent histone |
T3 | 307-324 | protein | denotes | homologue of Sir2 |
T4 | 326-331 | protein | denotes | SIRT1 |
T5 | 363-383 | protein | denotes | p53 tumor suppressor |
T6 | 412-416 | protein | denotes | Sir2 |
T7 | 800-804 | protein | denotes | Sir2 |
T8 | 895-899 | protein | denotes | Sir2 |
T9 | 998-1002 | protein | denotes | Sir2 |
T10 | 1007-1012 | protein | denotes | SIRT1 |
T11 | 1175-1183 | protein | denotes | proteins |
T12 | 1425-1437 | protein | denotes | Sir2 enzymes |
GlyCosmos15-HP
Id | Subject | Object | Predicate | Lexical cue | hp_id |
---|---|---|---|---|---|
T1 | 367-372 | Phenotype | denotes | tumor | HP:0002664 |
mondo_disease
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T1 | 367-372 | Disease | denotes | tumor | http://purl.obolibrary.org/obo/MONDO_0005070 |
NCBITAXON
Id | Subject | Object | Predicate | Lexical cue | db_id |
---|---|---|---|---|---|
T1 | 111-116 | OrganismTaxon | denotes | human | 9606 |
T2 | 128-152 | OrganismTaxon | denotes | Saccharomyces cerevisiae | 4932 |
T3 | 301-306 | OrganismTaxon | denotes | human | 9606 |