PubMed:12122014
Annnotations
PubTator4TogoVar
| Id | Subject | Object | Predicate | Lexical cue | proteinmutation |
|---|---|---|---|---|---|
| 12122014_0 | 794-799 | ProteinMutation | denotes | G129R | rs774669158 |
| 12122014_1 | 1011-1016 | ProteinMutation | denotes | G129R | rs774669158 |
| 12122014_2 | 1401-1406 | ProteinMutation | denotes | G129R | rs774669158 |
sentences
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-135 | Sentence | denotes | Csk homologous kinase (CHK) and ErbB-2 interactions are directly coupled with CHK negative growth regulatory function in breast cancer. |
| T2 | 136-394 | Sentence | denotes | Our previous studies demonstrated that Csk homologous kinase (CHK) acts as a negative growth regulator of human breast cancer through inhibition of ErbB-2/neu-mediated Src family kinase activity (Bougeret, C., Jiang, S., Keydar, I., and Avraham, H. (2001) J. |
| T3 | 395-400 | Sentence | denotes | Biol. |
| T4 | 401-406 | Sentence | denotes | Chem. |
| T5 | 407-424 | Sentence | denotes | 276, 33711-33720. |
| T6 | 425-568 | Sentence | denotes | The interaction between the CHK SH2 domain and Tyr(P)(1248) of the ErbB-2 receptor has been shown to be specific and critical for CHK function. |
| T7 | 569-740 | Sentence | denotes | In this report, we investigated whether the interaction of the CHK SH2 domain and ErbB-2 is directly related to the inhibition of heregulin-stimulated Src kinase activity. |
| T8 | 741-877 | Sentence | denotes | We constructed three CHK SH2 domain binding mutants: G129R (enhanced binding), R147K (inhibited binding), and R147A (disrupted binding). |
| T9 | 878-1010 | Sentence | denotes | NMR spectra for the domains of each construct were used to evaluate their interaction with a Tyr(P)(1248)-containing ErbB-2 peptide. |
| T10 | 1011-1102 | Sentence | denotes | G129R showed enhanced binding to ErbB-2, whereas binding was completely disrupted by R147A. |
| T11 | 1103-1290 | Sentence | denotes | The enhanced binding mutant showed chemical shift changes at the same residues as wild-type CHK, indicating that this mutant has the same binding characteristics as the wild-type protein. |
| T12 | 1291-1471 | Sentence | denotes | Furthermore, inhibition of heregulin-stimulated Src kinase activity was markedly diminished by R147A, whereas G129R-mediated inhibition was stronger as compared with wild-type CHK. |
| T13 | 1472-1629 | Sentence | denotes | These results indicate that the specific interaction of CHK and ErbB-2 via the SH2 domain of CHK is directly related to the growth inhibitory effects of CHK. |
| T14 | 1630-1801 | Sentence | denotes | These new CHK high affinity binding constructs may serve as good candidates for inhibition of the ErbB-2/Src transduction pathway in gene therapy studies in breast cancer. |
PubmedHPO
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 248-261 | HP_0003002 | denotes | breast cancer |
| T2 | 248-261 | HP_0100013 | denotes | breast cancer |
| T3 | 255-261 | HP_0002664 | denotes | cancer |
| T4 | 1787-1800 | HP_0003002 | denotes | breast cancer |
| T5 | 1787-1800 | HP_0100013 | denotes | breast cancer |
| T6 | 1794-1800 | HP_0002664 | denotes | cancer |
FSU-PRGE
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-21 | protein | denotes | Csk homologous kinase |
| T2 | 23-26 | protein | denotes | CHK |
| T3 | 32-38 | protein | denotes | ErbB-2 |
| T4 | 78-81 | protein | denotes | CHK |
| T5 | 175-196 | protein | denotes | Csk homologous kinase |
| T6 | 198-201 | protein | denotes | CHK |
| T7 | 284-290 | protein | denotes | ErbB-2 |
| T8 | 291-294 | protein | denotes | neu |
| T9 | 304-321 | protein | denotes | Src family kinase |
| T10 | 453-456 | protein | denotes | CHK |
| T11 | 492-498 | protein | denotes | ErbB-2 |
| T12 | 555-558 | protein | denotes | CHK |
| T13 | 632-635 | protein | denotes | CHK |
| T14 | 651-657 | protein | denotes | ErbB-2 |
| T15 | 699-708 | protein | denotes | heregulin |
| T16 | 720-730 | protein | denotes | Src kinase |
| T17 | 762-765 | protein | denotes | CHK |
| T18 | 995-1001 | protein | denotes | ErbB-2 |
| T19 | 1044-1050 | protein | denotes | ErbB-2 |
| T20 | 1195-1198 | protein | denotes | CHK |
| T21 | 1318-1327 | protein | denotes | heregulin |
| T22 | 1339-1349 | protein | denotes | Src kinase |
| T23 | 1467-1470 | protein | denotes | CHK |
| T24 | 1528-1531 | protein | denotes | CHK |
| T25 | 1536-1542 | protein | denotes | ErbB-2 |
| T26 | 1565-1568 | protein | denotes | CHK |
| T27 | 1625-1628 | protein | denotes | CHK |
| T28 | 1640-1643 | protein | denotes | CHK |
| T29 | 1728-1734 | protein | denotes | ErbB-2 |
| T30 | 1735-1738 | protein | denotes | Src |
PIR-corpus2
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-27 | protein | denotes | Csk homologous kinase (CHK) |
| T2 | 32-38 | protein | denotes | ErbB-2 |
| T3 | 78-81 | protein | denotes | CHK |
| T4 | 175-202 | protein | denotes | Csk homologous kinase (CHK) |
| T5 | 213-238 | protein | denotes | negative growth regulator |
| T6 | 284-290 | protein | denotes | ErbB-2 |
| T7 | 304-321 | protein | denotes | Src family kinase |
| T8 | 453-456 | protein | denotes | CHK |
| T9 | 492-498 | protein | denotes | ErbB-2 |
| T10 | 555-558 | protein | denotes | CHK |
| T11 | 632-635 | protein | denotes | CHK |
| T12 | 651-657 | protein | denotes | ErbB-2 |
| T13 | 699-719 | protein | denotes | heregulin-stimulated |
| T14 | 762-765 | protein | denotes | CHK |
| T15 | 995-1001 | protein | denotes | ErbB-2 |
| T16 | 1044-1050 | protein | denotes | ErbB-2 |
| T17 | 1195-1198 | protein | denotes | CHK |
| T18 | 1318-1349 | protein | denotes | heregulin-stimulated Src kinase |
| T19 | 1467-1470 | protein | denotes | CHK |
| T20 | 1528-1531 | protein | denotes | CHK |
| T21 | 1536-1542 | protein | denotes | ErbB-2 |
| T22 | 1565-1568 | protein | denotes | CHK |
| T23 | 1625-1628 | protein | denotes | CHK |
| T24 | 1640-1643 | protein | denotes | CHK |
| T25 | 1728-1734 | protein | denotes | ErbB-2 |
| T26 | 1735-1738 | protein | denotes | Src |
DisGeNET5_gene_disease
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| 12122014-0#0#21#gene4145 | 0-21 | gene4145 | denotes | Csk homologous kinase |
| 12122014-0#23#26#gene4145 | 23-26 | gene4145 | denotes | CHK |
| 12122014-0#32#38#gene2064 | 32-38 | gene2064 | denotes | ErbB-2 |
| 12122014-0#78#81#gene4145 | 78-81 | gene4145 | denotes | CHK |
| 12122014-0#121#134#diseaseC0006142 | 121-134 | diseaseC0006142 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0678222 | 121-134 | diseaseC0678222 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0006142 | 121-134 | diseaseC0006142 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0678222 | 121-134 | diseaseC0678222 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0006142 | 121-134 | diseaseC0006142 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0678222 | 121-134 | diseaseC0678222 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0006142 | 121-134 | diseaseC0006142 | denotes | breast cancer |
| 12122014-0#121#134#diseaseC0678222 | 121-134 | diseaseC0678222 | denotes | breast cancer |
| 0#21#gene4145121#134#diseaseC0006142 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0678222 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0006142 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0678222 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0006142 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0678222 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0006142 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | Csk homologous kinase,breast cancer |
| 0#21#gene4145121#134#diseaseC0678222 | 12122014-0#0#21#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | Csk homologous kinase,breast cancer |
| 23#26#gene4145121#134#diseaseC0006142 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0678222 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0006142 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0678222 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0006142 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0678222 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0006142 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 23#26#gene4145121#134#diseaseC0678222 | 12122014-0#23#26#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 32#38#gene2064121#134#diseaseC0006142 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0006142 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0678222 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0678222 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0006142 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0006142 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0678222 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0678222 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0006142 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0006142 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0678222 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0678222 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0006142 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0006142 | associated_with | ErbB-2,breast cancer |
| 32#38#gene2064121#134#diseaseC0678222 | 12122014-0#32#38#gene2064 | 12122014-0#121#134#diseaseC0678222 | associated_with | ErbB-2,breast cancer |
| 78#81#gene4145121#134#diseaseC0006142 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0678222 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0006142 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0678222 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0006142 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0678222 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0006142 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0006142 | associated_with | CHK,breast cancer |
| 78#81#gene4145121#134#diseaseC0678222 | 12122014-0#78#81#gene4145 | 12122014-0#121#134#diseaseC0678222 | associated_with | CHK,breast cancer |
PIR-corpus1
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-21 | protein | denotes | Csk homologous kinase |
| T2 | 23-26 | acronym | denotes | CHK |
| T3 | 32-38 | protein | denotes | ErbB-2 |
| T4 | 78-81 | protein | denotes | CHK |
| T5 | 175-196 | protein | denotes | Csk homologous kinase |
| T6 | 198-201 | acronym | denotes | CHK |
| T7 | 284-321 | protein | denotes | ErbB-2/neu-mediated Src family kinase |
| T8 | 492-498 | protein | denotes | ErbB-2 |
| T9 | 555-558 | protein | denotes | CHK |
| T10 | 651-657 | protein | denotes | ErbB-2 |
| T11 | 699-719 | protein | denotes | heregulin-stimulated |
| T12 | 1044-1050 | protein | denotes | ErbB-2 |
| T13 | 1195-1198 | protein | denotes | CHK |
| T14 | 1282-1289 | protein | denotes | protein |
| T15 | 1318-1349 | protein | denotes | heregulin-stimulated Src kinase |
| T16 | 1467-1470 | protein | denotes | CHK |
| T17 | 1528-1531 | protein | denotes | CHK |
| T18 | 1536-1542 | protein | denotes | ErbB-2 |
| T19 | 1565-1568 | protein | denotes | CHK |
| T20 | 1625-1628 | protein | denotes | CHK |
| T21 | 1728-1738 | protein | denotes | ErbB-2/Src |
DisGeNET
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T0 | 0-21 | gene:4145 | denotes | Csk homologous kinase |
| T1 | 121-134 | disease:C0006142 | denotes | breast cancer |
| T2 | 0-21 | gene:4145 | denotes | Csk homologous kinase |
| T3 | 121-134 | disease:C0678222 | denotes | breast cancer |
| T4 | 23-26 | gene:4145 | denotes | CHK |
| T5 | 121-134 | disease:C0006142 | denotes | breast cancer |
| T6 | 23-26 | gene:4145 | denotes | CHK |
| T7 | 121-134 | disease:C0678222 | denotes | breast cancer |
| T8 | 32-38 | gene:2064 | denotes | ErbB-2 |
| T9 | 121-134 | disease:C0006142 | denotes | breast cancer |
| T10 | 32-38 | gene:2064 | denotes | ErbB-2 |
| T11 | 121-134 | disease:C0678222 | denotes | breast cancer |
| T12 | 78-81 | gene:4145 | denotes | CHK |
| T13 | 121-134 | disease:C0678222 | denotes | breast cancer |
| T14 | 78-81 | gene:4145 | denotes | CHK |
| T15 | 121-134 | disease:C0006142 | denotes | breast cancer |
| T16 | 175-196 | gene:4145 | denotes | Csk homologous kinase |
| T17 | 248-261 | disease:C0006142 | denotes | breast cancer |
| T18 | 175-196 | gene:4145 | denotes | Csk homologous kinase |
| T19 | 248-261 | disease:C0678222 | denotes | breast cancer |
| T20 | 198-201 | gene:4145 | denotes | CHK |
| T21 | 248-261 | disease:C0006142 | denotes | breast cancer |
| T22 | 198-201 | gene:4145 | denotes | CHK |
| T23 | 248-261 | disease:C0678222 | denotes | breast cancer |
| R1 | T0 | T1 | associated_with | Csk homologous kinase,breast cancer |
| R2 | T2 | T3 | associated_with | Csk homologous kinase,breast cancer |
| R3 | T4 | T5 | associated_with | CHK,breast cancer |
| R4 | T6 | T7 | associated_with | CHK,breast cancer |
| R5 | T8 | T9 | associated_with | ErbB-2,breast cancer |
| R6 | T10 | T11 | associated_with | ErbB-2,breast cancer |
| R7 | T12 | T13 | associated_with | CHK,breast cancer |
| R8 | T14 | T15 | associated_with | CHK,breast cancer |
| R9 | T16 | T17 | associated_with | Csk homologous kinase,breast cancer |
| R10 | T18 | T19 | associated_with | Csk homologous kinase,breast cancer |
| R11 | T20 | T21 | associated_with | CHK,breast cancer |
| R12 | T22 | T23 | associated_with | CHK,breast cancer |
HP-phenotype
| Id | Subject | Object | Predicate | Lexical cue | hp_id |
|---|---|---|---|---|---|
| T1 | 121-134 | Phenotype | denotes | breast cancer | HP:0003002 |
| T2 | 248-261 | Phenotype | denotes | breast cancer | HP:0003002 |
| T3 | 1787-1800 | Phenotype | denotes | breast cancer | HP:0003002 |
mondo_disease
| Id | Subject | Object | Predicate | Lexical cue | mondo_id |
|---|---|---|---|---|---|
| T1 | 121-134 | Disease | denotes | breast cancer | http://purl.obolibrary.org/obo/MONDO_0007254 |
| T2 | 248-261 | Disease | denotes | breast cancer | http://purl.obolibrary.org/obo/MONDO_0007254 |
| T3 | 1787-1800 | Disease | denotes | breast cancer | http://purl.obolibrary.org/obo/MONDO_0007254 |
NCBITAXON
| Id | Subject | Object | Predicate | Lexical cue | db_id |
|---|---|---|---|---|---|
| T1 | 242-247 | OrganismTaxon | denotes | human | 9606 |
Anatomy-UBERON
| Id | Subject | Object | Predicate | Lexical cue | uberon_id |
|---|---|---|---|---|---|
| T1 | 121-127 | Body_part | denotes | breast | http://purl.obolibrary.org/obo/UBERON_0000310 |
| T2 | 248-254 | Body_part | denotes | breast | http://purl.obolibrary.org/obo/UBERON_0000310 |
| T3 | 1787-1793 | Body_part | denotes | breast | http://purl.obolibrary.org/obo/UBERON_0000310 |