PubMed:10217534
Annnotations
PMID_GLOBAL
| Id | Subject | Object | Predicate | Lexical cue | mondo_id |
|---|---|---|---|---|---|
| T1 | 80-96 | DiseaseOrPhenotypicFeature | denotes | hypersensitivity | 0000605|0005271 |
| T3 | 245-261 | DiseaseOrPhenotypicFeature | denotes | hypersensitivity | 0000605|0005271 |
| T5 | 1210-1219 | DiseaseOrPhenotypicFeature | denotes | sensitive | 0000605 |
| T6 | 1677-1680 | DiseaseOrPhenotypicFeature | denotes | can | 0012833 |
| T7 | 1711-1727 | DiseaseOrPhenotypicFeature | denotes | hypersensitivity | 0000605|0005271 |
jnlpba-st-training
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 528-545 | cell_type | denotes | white blood cells |
| T2 | 718-746 | cell_type | denotes | human peripheral blood cells |
| T3 | 800-810 | protein | denotes | ubiquitous |
| T4 | 1165-1176 | cell_type | denotes | Lymphocytes |
| T5 | 1267-1278 | cell_type | denotes | neutrophils |
| T6 | 1313-1328 | cell_type | denotes | red blood cells |
pubmed-sentences-benchmark
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| S1 | 0-97 | Sentence | denotes | Cellular disposition of sulphamethoxazole and its metabolites: implications for hypersensitivity. |
| S2 | 98-262 | Sentence | denotes | 1. Bioactivation of sulphamethoxazole (SMX) to chemically-reactive metabolites and subsequent protein conjugation is thought to be involved in SMX hypersensitivity. |
| S3 | 263-379 | Sentence | denotes | We have therefore examined the cellular metabolism, disposition and conjugation of SMX and its metabolites in vitro. |
| S4 | 380-546 | Sentence | denotes | 2. Flow cytometry revealed binding of N-hydroxy (SMX-NHOH) and nitroso (SMX-NO) metabolites of SMX, but not of SMX itself, to the surface of viable white blood cells. |
| S5 | 547-621 | Sentence | denotes | Cellular haptenation by SMX-NO was reduced by exogenous glutathione (GSH). |
| S6 | 622-837 | Sentence | denotes | 3. SMX-NHOH and SMX-NO were rapidly reduced back to the parent compound by cysteine (CYS), GSH, human peripheral blood cells and plasma, suggesting that this is an important and ubiquitous bioinactivation mechanism. |
| S7 | 838-967 | Sentence | denotes | 4. Fluorescence HPLC showed that SMX-NHOH and SMX-NO depleted CYS and GSH in buffer, and to a lesser extent, in cells and plasma. |
| S8 | 968-1164 | Sentence | denotes | 5. Neutrophil apoptosis and inhibition of neutrophil function were induced at lower concentrations of SMX-NHOH and SMX-NO than those inducing loss of membrane viability, with SMX having no effect. |
| S9 | 1165-1279 | Sentence | denotes | Lymphocytes were significantly (P<0.05) more sensitive to the direct cytotoxic effects of SMX-NO than neutrophils. |
| S10 | 1280-1401 | Sentence | denotes | 6. Partitioning of SMX-NHOH into red blood cells was significantly (P<0.05) lower than with the hydroxylamine of dapsone. |
| S11 | 1402-1558 | Sentence | denotes | 7. Our results suggest that the balance between oxidation of SMX to its toxic metabolites and their reduction is an important protective cellular mechanism. |
| S12 | 1559-1728 | Sentence | denotes | If an imbalance exists, haptenation of the toxic metabolites to bodily proteins including the surface of viable cells can occur, and may result in drug hypersensitivity. |
genia-medco-coref
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| C2 | 24-41 | NP | denotes | sulphamethoxazole |
| C3 | 46-49 | NP | denotes | its |
| C1 | 24-61 | NP | denotes | sulphamethoxazole and its metabolites |
| C4 | 118-141 | NP | denotes | sulphamethoxazole (SMX) |
| C6 | 346-349 | NP | denotes | SMX |
| C7 | 354-357 | NP | denotes | its |
| C5 | 346-369 | NP | denotes | SMX and its metabolites |
| C9 | 475-478 | NP | denotes | SMX |
| C8 | 418-478 | NP | denotes | N-hydroxy (SMX-NHOH) and nitroso (SMX-NO) metabolites of SMX |
| C10 | 491-501 | NP | denotes | SMX itself |
| C11 | 571-577 | NP | denotes | SMX-NO |
| C12 | 593-620 | NP | denotes | exogenous glutathione (GSH) |
| C14 | 625-633 | NP | denotes | SMX-NHOH |
| C15 | 638-644 | NP | denotes | SMX-NO |
| C13 | 625-644 | NP | denotes | SMX-NHOH and SMX-NO |
| C16 | 713-716 | NP | denotes | GSH |
| C17 | 751-757 | NP | denotes | plasma |
| C19 | 871-879 | NP | denotes | SMX-NHOH |
| C20 | 884-890 | NP | denotes | SMX-NO |
| C18 | 871-890 | NP | denotes | SMX-NHOH and SMX-NO |
| C21 | 960-966 | NP | denotes | plasma |
| C23 | 1070-1078 | NP | denotes | SMX-NHOH |
| C24 | 1083-1089 | NP | denotes | SMX-NO |
| C22 | 1070-1089 | NP | denotes | SMX-NHOH and SMX-NO |
| C25 | 1255-1261 | NP | denotes | SMX-NO |
| C26 | 1299-1307 | NP | denotes | SMX-NHOH |
| C27 | 1463-1466 | NP | denotes | SMX |
| C29 | 1470-1473 | NP | denotes | its |
| C28 | 1470-1491 | NP | denotes | its toxic metabolites |
| C30 | 1496-1501 | NP | denotes | their |
| C31 | 1598-1619 | NP | denotes | the toxic metabolites |
| R1 | C3 | C2 | coref-pron | its,sulphamethoxazole |
| R2 | C4 | C2 | coref-ident | sulphamethoxazole (SMX),sulphamethoxazole |
| R3 | C6 | C4 | coref-ident | SMX,sulphamethoxazole (SMX) |
| R4 | C7 | C6 | coref-pron | its,SMX |
| R5 | C5 | C1 | coref-ident | SMX and its metabolites,sulphamethoxazole and its metabolites |
| R6 | C9 | C6 | coref-ident | SMX,SMX |
| R7 | C10 | C9 | coref-ident | SMX itself,SMX |
| R8 | C15 | C11 | coref-ident | SMX-NO,SMX-NO |
| R9 | C13 | C8 | coref-ident | SMX-NHOH and SMX-NO,N-hydroxy (SMX-NHOH) and nitroso (SMX-NO) metabolites of SMX |
| R10 | C16 | C12 | coref-ident | GSH,exogenous glutathione (GSH) |
| R11 | C19 | C14 | coref-ident | SMX-NHOH,SMX-NHOH |
| R12 | C20 | C15 | coref-ident | SMX-NO,SMX-NO |
| R13 | C18 | C13 | coref-ident | SMX-NHOH and SMX-NO,SMX-NHOH and SMX-NO |
| R14 | C21 | C17 | coref-ident | plasma,plasma |
| R15 | C23 | C19 | coref-ident | SMX-NHOH,SMX-NHOH |
| R16 | C24 | C20 | coref-ident | SMX-NO,SMX-NO |
| R17 | C22 | C18 | coref-ident | SMX-NHOH and SMX-NO,SMX-NHOH and SMX-NO |
| R18 | C25 | C24 | coref-ident | SMX-NO,SMX-NO |
| R19 | C26 | C23 | coref-ident | SMX-NHOH,SMX-NHOH |
| R20 | C27 | C10 | coref-ident | SMX,SMX itself |
| R21 | C29 | C27 | coref-pron | its,SMX |
| R22 | C30 | C28 | coref-pron | their,its toxic metabolites |
| R23 | C31 | C28 | coref-ident | the toxic metabolites,its toxic metabolites |
GENIAcorpus
| Id | Subject | Object | Predicate | Lexical cue |
|---|---|---|---|---|
| T1 | 0-20 | other_name | denotes | Cellular disposition |
| T2 | 24-41 | other_organic_compound | denotes | sulphamethoxazole |
| T3 | 50-61 | other_organic_compound | denotes | metabolites |
| T4 | 63-96 | other_name | denotes | implications for hypersensitivity |
| T5 | 118-135 | other_organic_compound | denotes | sulphamethoxazole |
| T6 | 137-140 | other_organic_compound | denotes | SMX |
| T7 | 165-176 | other_organic_compound | denotes | metabolites |
| T8 | 192-211 | other_name | denotes | protein conjugation |
| T9 | 241-244 | other_organic_compound | denotes | SMX |
| T10 | 346-349 | other_organic_compound | denotes | SMX |
| T11 | 358-369 | other_organic_compound | denotes | metabolites |
| T12 | 475-478 | other_organic_compound | denotes | SMX |
| T13 | 491-494 | other_organic_compound | denotes | SMX |
| T14 | 528-545 | cell_type | denotes | white blood cells |
| T15 | 571-574 | other_organic_compound | denotes | SMX |
| T16 | 603-614 | peptide | denotes | glutathione |
| T17 | 616-619 | peptide | denotes | GSH |
| T18 | 625-628 | other_organic_compound | denotes | SMX |
| T19 | 638-641 | other_organic_compound | denotes | SMX |
| T20 | 697-705 | amino_acid_monomer | denotes | cysteine |
| T21 | 707-710 | amino_acid_monomer | denotes | CYS |
| T22 | 713-716 | peptide | denotes | GSH |
| T23 | 718-746 | cell_type | denotes | human peripheral blood cells |
| T24 | 800-810 | protein_family_or_group | denotes | ubiquitous |
| T25 | 841-858 | other_name | denotes | Fluorescence HPLC |
| T26 | 871-874 | other_organic_compound | denotes | SMX |
| T27 | 884-887 | other_organic_compound | denotes | SMX |
| T28 | 900-903 | amino_acid_monomer | denotes | CYS |
| T29 | 908-911 | peptide | denotes | GSH |
| T30 | 960-966 | tissue | denotes | plasma |
| T31 | 971-991 | other_name | denotes | Neutrophil apoptosis |
| T32 | 1010-1029 | other_name | denotes | neutrophil function |
| T33 | 1070-1073 | other_organic_compound | denotes | SMX |
| T34 | 1083-1086 | other_organic_compound | denotes | SMX |
| T35 | 1143-1146 | other_organic_compound | denotes | SMX |
| T36 | 1165-1176 | cell_type | denotes | Lymphocytes |
| T37 | 1234-1251 | other_name | denotes | cytotoxic effects |
| T38 | 1255-1258 | other_organic_compound | denotes | SMX |
| T39 | 1267-1278 | cell_type | denotes | neutrophils |
| T40 | 1299-1302 | other_organic_compound | denotes | SMX |
| T41 | 1313-1328 | cell_type | denotes | red blood cells |
| T42 | 1376-1389 | other_organic_compound | denotes | hydroxylamine |
| T43 | 1393-1400 | other_organic_compound | denotes | dapsone |
| T44 | 1463-1466 | other_organic_compound | denotes | SMX |
| T45 | 1583-1594 | other_name | denotes | haptenation |
| T46 | 1602-1619 | other_organic_compound | denotes | toxic metabolites |
| T47 | 1706-1727 | other_name | denotes | drug hypersensitivity |