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PMC:7461420 / 38656-39463
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T203 | 467-474 | Body_part | denotes | leucine | http://purl.org/sig/ont/fma/fma82757 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T210 | 53-57 | Disease | denotes | SARS | http://purl.obolibrary.org/obo/MONDO_0005091 |
T211 | 300-337 | Disease | denotes | porcine transmissible gastroenteritis | http://purl.obolibrary.org/obo/MONDO_0025420 |
T212 | 322-337 | Disease | denotes | gastroenteritis | http://purl.obolibrary.org/obo/MONDO_0002269 |
T213 | 517-521 | Disease | denotes | SARS | http://purl.obolibrary.org/obo/MONDO_0005091 |
T214 | 780-784 | Disease | denotes | SARS | http://purl.obolibrary.org/obo/MONDO_0005091 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T452 | 85-86 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T453 | 87-95 | http://purl.obolibrary.org/obo/PR_000018263 | denotes | peptidic |
T454 | 110-113 | http://purl.obolibrary.org/obo/CLO_0037067 | denotes | Val |
T455 | 273-274 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T456 | 365-366 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T457 | 398-400 | http://purl.obolibrary.org/obo/CLO_0008285 | denotes | P1 |
T458 | 440-442 | http://purl.obolibrary.org/obo/CLO_0050050 | denotes | S1 |
T459 | 464-466 | http://purl.obolibrary.org/obo/CLO_0008307 | denotes | P2 |
T460 | 506-508 | http://purl.obolibrary.org/obo/CLO_0008922 | denotes | S2 |
T461 | 506-508 | http://purl.obolibrary.org/obo/CLO_0050052 | denotes | S2 |
T462 | 574-575 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T463 | 604-609 | http://purl.obolibrary.org/obo/NCBITaxon_9606 | denotes | human |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T356 | 96-105 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T357 | 106-109 | Chemical | denotes | Cbz | http://purl.obolibrary.org/obo/CHEBI_51097 |
T358 | 110-113 | Chemical | denotes | Val | http://purl.obolibrary.org/obo/CHEBI_16414|http://purl.obolibrary.org/obo/CHEBI_30015 |
T360 | 114-117 | Chemical | denotes | Asn | http://purl.obolibrary.org/obo/CHEBI_17196|http://purl.obolibrary.org/obo/CHEBI_22653|http://purl.obolibrary.org/obo/CHEBI_50347 |
T363 | 118-121 | Chemical | denotes | Ser | http://purl.obolibrary.org/obo/CHEBI_17115|http://purl.obolibrary.org/obo/CHEBI_29999 |
T365 | 122-125 | Chemical | denotes | Thr | http://purl.obolibrary.org/obo/CHEBI_16857|http://purl.obolibrary.org/obo/CHEBI_30013 |
T367 | 126-129 | Chemical | denotes | Leu | http://purl.obolibrary.org/obo/CHEBI_15603|http://purl.obolibrary.org/obo/CHEBI_25017|http://purl.obolibrary.org/obo/CHEBI_30006 |
T370 | 130-133 | Chemical | denotes | Gln | http://purl.obolibrary.org/obo/CHEBI_30011 |
T371 | 147-153 | Chemical | denotes | ketone | http://purl.obolibrary.org/obo/CHEBI_17087 |
T372 | 194-200 | Chemical | denotes | ketone | http://purl.obolibrary.org/obo/CHEBI_17087 |
T373 | 398-400 | Chemical | denotes | P1 | http://purl.obolibrary.org/obo/CHEBI_60949 |
T374 | 401-404 | Chemical | denotes | Gln | http://purl.obolibrary.org/obo/CHEBI_30011 |
T375 | 464-466 | Chemical | denotes | P2 | http://purl.obolibrary.org/obo/CHEBI_33472 |
T376 | 467-474 | Chemical | denotes | leucine | http://purl.obolibrary.org/obo/CHEBI_25017 |
T377 | 506-508 | Chemical | denotes | S2 | http://purl.obolibrary.org/obo/CHEBI_29387 |
T378 | 576-590 | Chemical | denotes | peptidomimetic | http://purl.obolibrary.org/obo/CHEBI_63175 |
T379 | 591-600 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T380 | 656-665 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T381 | 720-729 | Chemical | denotes | molecules | http://purl.obolibrary.org/obo/CHEBI_25367 |
T382 | 791-806 | Chemical | denotes | Mpro inhibitors | http://purl.obolibrary.org/obo/CHEBI_147285 |
T383 | 796-806 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
1200 | 791-795 | Gene | denotes | Mpro | Gene:8673700 |
1201 | 64-68 | Gene | denotes | Mpro | Gene:8673700 |
1202 | 699-703 | Gene | denotes | Mpro | Gene:8673700 |
1203 | 528-532 | Gene | denotes | Mpro | Gene:8673700 |
1204 | 349-353 | Gene | denotes | Mpro | Gene:8673700 |
1205 | 53-61 | Species | denotes | SARS‐CoV | Tax:694009 |
1206 | 343-347 | Species | denotes | TGEV | Tax:11149 |
1207 | 517-525 | Species | denotes | SARS‐CoV | Tax:694009 |
1208 | 604-622 | Species | denotes | human rhinovirus 3 | Tax:44130 |
1209 | 694-698 | Species | denotes | TGEV | Tax:11149 |
1210 | 780-788 | Species | denotes | SARS‐CoV | Tax:694009 |
1211 | 308-321 | Species | denotes | transmissible | Tax:11149 |
1212 | 106-153 | Chemical | denotes | Cbz‐Val‐Asn‐Ser‐Thr‐Leu‐Gln‐chloromethyl ketone | |
1213 | 181-200 | Chemical | denotes | chloromethyl ketone | |
1214 | 398-400 | Chemical | denotes | P1 | MESH:C480041 |
1215 | 401-404 | Chemical | denotes | Gln | MESH:D005973 |
1216 | 467-474 | Chemical | denotes | leucine | MESH:D007930 |
1217 | 548-559 | Chemical | denotes | rupintrivir | MESH:C118874 |
1218 | 565-571 | Chemical | denotes | AG7088 | MESH:C118874 |
1219 | 322-341 | Disease | denotes | gastroenteritis CoV | MESH:C000657245 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T358 | 0-257 | Sentence | denotes | The disclosure of the first crystal structure of the SARS‐CoV‐1 Mpro in complex with a peptidic inhibitor Cbz‐Val‐Asn‐Ser‐Thr‐Leu‐Gln‐chloromethyl ketone (also known as hexapeptide chloromethyl ketone; 28) 125 provided clues for the substrate‐based design. |
T359 | 258-533 | Sentence | denotes | Although it is a substrate analog for the porcine transmissible gastroenteritis CoV (TGEV) Mpro, it offers a structural explanation for the P1‐Gln entering into the specific subsite S1 pocket and decreased P2‐leucine specificity in the hydrophobic S2 site of SARS‐CoV‐1 Mpro. |
T360 | 534-704 | Sentence | denotes | Additionally, rupintrivir (29; AG7088), a peptidomimetic inhibitor of human rhinovirus 3C protease is oriented similar to inhibitor 28 in the binding pocket of TGEV Mpro. |
T361 | 705-807 | Sentence | denotes | 129 These two molecules became prototype compounds for the development of SARS‐CoV‐1 Mpro inhibitors. |