
PMC:7291971 / 44379-45856
Annnotations
LitCovid-PMC-OGER-BB
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T926 | 9-11 | CHEBI:53424;CHEBI:53424 | denotes | 22 |
T927 | 93-98 | CHEBI:15377;CHEBI:15377 | denotes | water |
T928 | 133-141 | CHEBI:46787;CHEBI:46787 | denotes | solvents |
T929 | 198-203 | CHEBI:15377;CHEBI:15377 | denotes | water |
T930 | 221-228 | CHEBI:15377;CHEBI:15377 | denotes | aqueous |
T931 | 229-233 | CHEBI:48607;CHEBI:48607 | denotes | LiOH |
T932 | 234-242 | CHEBI:75958;CHEBI:75958 | denotes | solution |
T933 | 340-347 | CHEBI:15377;CHEBI:15377 | denotes | aqueous |
T934 | 348-351 | CHEBI:17883;CHEBI:17883 | denotes | HCl |
T935 | 352-360 | CHEBI:75958;CHEBI:75958 | denotes | solution |
T936 | 366-373 | CHEBI:46787;CHEBI:46787 | denotes | solvent |
T937 | 479-485 | CHEBI:30563;CHEBI:30563 | denotes | silica |
T938 | 546-558 | CHEBI:38472;CHEBI:38472 | denotes | acetonitrile |
T939 | 622-630 | CHEBI:36357;CHEBI:36357 | denotes | compound |
T940 | 678-683 | CHEBI:15377;CHEBI:15377 | denotes | water |
T941 | 1215-1218 | CHEBI:36927;CHEBI:36927 | denotes | 13C |
T17648 | 9-11 | CHEBI:53424;CHEBI:53424 | denotes | 22 |
T7216 | 93-98 | CHEBI:15377;CHEBI:15377 | denotes | water |
T10240 | 133-141 | CHEBI:46787;CHEBI:46787 | denotes | solvents |
T70971 | 198-203 | CHEBI:15377;CHEBI:15377 | denotes | water |
T82680 | 221-228 | CHEBI:15377;CHEBI:15377 | denotes | aqueous |
T99687 | 229-233 | CHEBI:48607;CHEBI:48607 | denotes | LiOH |
T12422 | 234-242 | CHEBI:75958;CHEBI:75958 | denotes | solution |
T45037 | 340-347 | CHEBI:15377;CHEBI:15377 | denotes | aqueous |
T26603 | 348-351 | CHEBI:17883;CHEBI:17883 | denotes | HCl |
T15792 | 352-360 | CHEBI:75958;CHEBI:75958 | denotes | solution |
T22239 | 366-373 | CHEBI:46787;CHEBI:46787 | denotes | solvent |
T42331 | 479-485 | CHEBI:30563;CHEBI:30563 | denotes | silica |
T43871 | 546-558 | CHEBI:38472;CHEBI:38472 | denotes | acetonitrile |
T83104 | 622-630 | CHEBI:36357;CHEBI:36357 | denotes | compound |
T77066 | 678-683 | CHEBI:15377;CHEBI:15377 | denotes | water |
T3324 | 1215-1218 | CHEBI:36927;CHEBI:36927 | denotes | 13C |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
792 | 77-80 | Chemical | denotes | TFA | MESH:D014269 |
793 | 93-98 | Chemical | denotes | water | MESH:D014867 |
794 | 198-203 | Chemical | denotes | water | MESH:D014867 |
795 | 229-233 | Chemical | denotes | LiOH | |
796 | 348-351 | Chemical | denotes | HCl | MESH:D006851 |
797 | 479-485 | Chemical | denotes | silica | MESH:D012822 |
798 | 497-500 | Chemical | denotes | C18 | MESH:C109760 |
799 | 546-558 | Chemical | denotes | acetonitrile | MESH:C032159 |
800 | 562-567 | Chemical | denotes | TEAAc | |
801 | 678-683 | Chemical | denotes | water | MESH:D014867 |
802 | 1215-1218 | Chemical | denotes | 13C | MESH:C000615229 |
803 | 1233-1236 | Chemical | denotes | D2O | |
804 | 1431-1442 | Chemical | denotes | C26H37N12O9 | |
805 | 1404-1408 | Disease | denotes | HRMS |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T308 | 9-11 | http://purl.obolibrary.org/obo/CLO_0050507 | denotes | 22 |
T309 | 462-463 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T310 | 519-520 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T311 | 710-711 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T312 | 1444-1447 | http://purl.obolibrary.org/obo/CLO_0007706 | denotes | M+H |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T812 | 77-80 | Chemical | denotes | TFA | http://purl.obolibrary.org/obo/CHEBI_45892 |
T813 | 93-98 | Chemical | denotes | water | http://purl.obolibrary.org/obo/CHEBI_15377 |
T814 | 133-141 | Chemical | denotes | solvents | http://purl.obolibrary.org/obo/CHEBI_46787 |
T815 | 198-203 | Chemical | denotes | water | http://purl.obolibrary.org/obo/CHEBI_15377 |
T816 | 229-233 | Chemical | denotes | LiOH | http://purl.obolibrary.org/obo/CHEBI_33979 |
T817 | 234-242 | Chemical | denotes | solution | http://purl.obolibrary.org/obo/CHEBI_75958 |
T818 | 348-351 | Chemical | denotes | HCl | http://purl.obolibrary.org/obo/CHEBI_17883 |
T819 | 352-360 | Chemical | denotes | solution | http://purl.obolibrary.org/obo/CHEBI_75958 |
T820 | 366-373 | Chemical | denotes | solvent | http://purl.obolibrary.org/obo/CHEBI_46787 |
T821 | 479-485 | Chemical | denotes | silica | http://purl.obolibrary.org/obo/CHEBI_30563 |
T822 | 546-558 | Chemical | denotes | acetonitrile | http://purl.obolibrary.org/obo/CHEBI_38472 |
T823 | 568-574 | Chemical | denotes | buffer | http://purl.obolibrary.org/obo/CHEBI_35225 |
T824 | 678-683 | Chemical | denotes | water | http://purl.obolibrary.org/obo/CHEBI_15377 |
T825 | 780-782 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T826 | 797-800 | Chemical | denotes | D2O | http://purl.obolibrary.org/obo/CHEBI_41981 |
T827 | 813-815 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T828 | 827-829 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T829 | 841-843 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T830 | 855-857 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T831 | 881-883 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T832 | 907-909 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T833 | 965-967 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T834 | 984-986 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T835 | 1043-1045 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T836 | 1099-1101 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T837 | 1164-1166 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T838 | 1191-1193 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T839 | 1233-1236 | Chemical | denotes | D2O | http://purl.obolibrary.org/obo/CHEBI_41981 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T324 | 0-108 | Sentence | denotes | Compound 22 (86 mg, 75.3 μmol, 1.00 eq) was treated at room temperature with TFA (830 μL) in water (210 μL). |
T325 | 109-168 | Sentence | denotes | After stirring for 3 h, solvents were removed under vacuum. |
T326 | 169-260 | Sentence | denotes | The residue was dissolved in water (0.5 mL) and 2 M aqueous LiOH solution (4 mL) was added. |
T327 | 261-361 | Sentence | denotes | After stirring at 0 °C for 30 min, pH ≈ 3 or 4 was adjusted by addition of 1 M aqueous HCl solution. |
T328 | 362-587 | Sentence | denotes | The solvent was removed under vacuum and the residue was purified by flash column chromatography on a reversed-phase silica gel column C18 (4 g, 40 μm) with a 0–15% linear gradient of acetonitrile in TEAAc buffer 50 mM, pH 7. |
T329 | 588-779 | Sentence | denotes | The fractions containing the pure compound were pooled, concentrated and lyophilized with water to give 2 (16 mg, 32%) as a white powder with 99% purity determined by HPLC analysis at 260 nm. |
T330 | 780-1214 | Sentence | denotes | 1H NMR (600 MHz, D2O) δ 8.11 (s, 1H), 8.05 (s, 1H), 7.98 (s, 1H), 7.86 (s, 1H), 5.89 (d, J = 2.5 Hz, 1H), 5.77 (d, J = 3.3 Hz, 1H), 4.51–4.47 (m, 2H), 4.36 (dd, J = 5.1 Hz, J = 3.4 Hz, 1H), 4.34–4.29 (m, 1H), 4.14–4.08 (m, 2H), 3.97 (td, J = 10.6 Hz, J = 2.4 Hz, 1H), 3.89–3.80 (m, 3H), 3.71 (dd, J = 13.0, J = 3.4 Hz, 1H), 3.15–3.04 (m, 2H), 3.03–2.81 (m, 2H), 2.76 (d, J = 14.2 Hz, 1H), 2.58 (d, J = 13.8 Hz, 1H), 2.14–1.99 (m, 2H). |
T331 | 1215-1403 | Sentence | denotes | 13C NMR (150 MHz, D2O) δ 174.5, 154.9 (2C) 152.5, 152.2, 147.7, 147.5, 139.3, 138.5, 118.5, 118.2, 89.0, 86.8, 84.8, 81.7, 80.0, 73.9, 71.1, 68.9, 67.7, 60.3, 56.2, 55.3, 53.8, 52.5, 26.1. |
T332 | 1404-1450 | Sentence | denotes | HRMS (ESI+): m/z calcd for C26H37N12O9 [M+H]+: |
T333 | 1451-1467 | Sentence | denotes | 661.2806, found: |
T334 | 1468-1477 | Sentence | denotes | 661.2811. |