PMC:7102591 / 26561-28716
Annnotations
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
829 | 198-220 | Gene | denotes | numb-associated kinase | Gene:29110 |
830 | 222-225 | Gene | denotes | NAK | Gene:29110 |
831 | 243-274 | Gene | denotes | AP2-associated protein kinase 1 | Gene:22848 |
832 | 276-280 | Gene | denotes | AAK1 | Gene:22848 |
833 | 286-312 | Gene | denotes | cyclin G-associated kinase | Gene:2580 |
834 | 314-317 | Gene | denotes | GAK | Gene:2580 |
835 | 340-344 | Gene | denotes | AAK1 | Gene:22848 |
836 | 462-466 | Gene | denotes | AAK1 | Gene:22848 |
837 | 512-516 | Gene | denotes | AAK1 | Gene:22848 |
838 | 823-826 | Gene | denotes | NAK | Gene:29110 |
839 | 1051-1055 | Gene | denotes | AAK1 | Gene:22848 |
840 | 1060-1063 | Gene | denotes | GAK | Gene:2580 |
841 | 1213-1224 | Gene | denotes | JAK 1 and 2 | Gene:3716 |
842 | 1337-1341 | Gene | denotes | IL-6 | Gene:3569 |
843 | 1758-1762 | Gene | denotes | AAK1 | Gene:22848 |
844 | 1346-1362 | Gene | denotes | interferon gamma | Gene:3458 |
845 | 35-45 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
846 | 693-705 | Species | denotes | Dengue virus | Tax:12637 |
847 | 707-718 | Species | denotes | Ebola virus | Tax:205488 |
848 | 724-751 | Species | denotes | respiratory syncytial virus | Tax:12814 |
849 | 959-966 | Species | denotes | patient | Tax:9606 |
850 | 576-585 | Chemical | denotes | erlotinib | MESH:D000069347 |
851 | 587-596 | Chemical | denotes | sunitinib | MESH:D000077210 |
852 | 598-609 | Chemical | denotes | ruxolitinib | MESH:C540383 |
853 | 615-625 | Chemical | denotes | fedratinib | MESH:C528327 |
854 | 1008-1019 | Chemical | denotes | baricitinib | MESH:C000596027 |
855 | 1226-1237 | Chemical | denotes | baricitinib | MESH:C000596027 |
856 | 1491-1502 | Chemical | denotes | baricitinib | MESH:C000596027 |
857 | 1655-1674 | Chemical | denotes | lopinavir/ritonavir | MESH:C558899 |
858 | 1679-1689 | Chemical | denotes | remdesivir | MESH:C000606551 |
859 | 1712-1723 | Chemical | denotes | tofacitinib | MESH:C479163 |
860 | 1892-1904 | Chemical | denotes | upadacitinib | MESH:C000613732 |
861 | 1908-1918 | Chemical | denotes | filgotinib | MESH:C584571 |
862 | 2124-2135 | Chemical | denotes | ruxolitinib | MESH:C540383 |
863 | 671-680 | Disease | denotes | infection | MESH:D007239 |
864 | 1147-1149 | Disease | denotes | RA | MESH:D001172 |
865 | 1418-1427 | Disease | denotes | pneumonia | MESH:D011014 |
866 | 1435-1443 | Disease | denotes | COVID-19 | MESH:C000657245 |
867 | 1880-1882 | Disease | denotes | RA | MESH:D001172 |
868 | 1935-1956 | Disease | denotes | coronavirus infection | MESH:D018352 |
869 | 2089-2097 | Disease | denotes | COVID-19 | MESH:C000657245 |
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T100 | 62-67 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T101 | 149-157 | Body_part | denotes | clathrin | http://purl.org/sig/ont/fma/fma62262 |
T102 | 258-265 | Body_part | denotes | protein | http://purl.org/sig/ont/fma/fma67257 |
T103 | 383-387 | Body_part | denotes | lung | http://purl.org/sig/ont/fma/fma7195 |
T104 | 388-393 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T105 | 684-689 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T106 | 1071-1077 | Body_part | denotes | plasma | http://purl.org/sig/ont/fma/fma62970 |
T107 | 2029-2037 | Body_part | denotes | clathrin | http://purl.org/sig/ont/fma/fma62262 |
LitCovid-PD-UBERON
Id | Subject | Object | Predicate | Lexical cue | uberon_id |
---|---|---|---|---|---|
T28 | 383-387 | Body_part | denotes | lung | http://purl.obolibrary.org/obo/UBERON_0002048 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T290 | 35-43 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T291 | 671-680 | Disease | denotes | infection | http://purl.obolibrary.org/obo/MONDO_0005550 |
T292 | 693-699 | Disease | denotes | Dengue | http://purl.obolibrary.org/obo/MONDO_0005502 |
T293 | 707-712 | Disease | denotes | Ebola | http://purl.obolibrary.org/obo/MONDO_0005737 |
T294 | 1147-1149 | Disease | denotes | RA | http://purl.obolibrary.org/obo/MONDO_0005272|http://purl.obolibrary.org/obo/MONDO_0008383 |
T296 | 1322-1325 | Disease | denotes | CRS | http://purl.obolibrary.org/obo/MONDO_0007399|http://purl.obolibrary.org/obo/MONDO_0017361 |
T298 | 1418-1427 | Disease | denotes | pneumonia | http://purl.obolibrary.org/obo/MONDO_0005249 |
T299 | 1435-1443 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
T300 | 1880-1882 | Disease | denotes | RA | http://purl.obolibrary.org/obo/MONDO_0005272|http://purl.obolibrary.org/obo/MONDO_0008383 |
T302 | 1947-1956 | Disease | denotes | infection | http://purl.obolibrary.org/obo/MONDO_0005550 |
T303 | 2089-2097 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T200 | 62-67 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T201 | 314-317 | http://purl.obolibrary.org/obo/CLO_0037126 | denotes | GAK |
T202 | 372-377 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T203 | 383-387 | http://purl.obolibrary.org/obo/UBERON_0002048 | denotes | lung |
T204 | 383-387 | http://www.ebi.ac.uk/efo/EFO_0000934 | denotes | lung |
T205 | 388-393 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T206 | 433-438 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T207 | 450-453 | http://purl.obolibrary.org/obo/CLO_0054060 | denotes | 102 |
T208 | 684-689 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T209 | 700-705 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T210 | 713-718 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T211 | 746-751 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T212 | 1060-1063 | http://purl.obolibrary.org/obo/CLO_0037126 | denotes | GAK |
T213 | 1071-1077 | http://purl.obolibrary.org/obo/UBERON_0001969 | denotes | plasma |
T214 | 1188-1189 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T215 | 1346-1362 | http://purl.obolibrary.org/obo/PR_000000017 | denotes | interferon gamma |
T216 | 1566-1567 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T217 | 1869-1875 | http://purl.obolibrary.org/obo/UBERON_0000473 | denotes | tested |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T213 | 258-265 | Chemical | denotes | protein | http://purl.obolibrary.org/obo/CHEBI_36080 |
T214 | 576-585 | Chemical | denotes | erlotinib | http://purl.obolibrary.org/obo/CHEBI_114785 |
T215 | 587-596 | Chemical | denotes | sunitinib | http://purl.obolibrary.org/obo/CHEBI_38940 |
T216 | 598-609 | Chemical | denotes | ruxolitinib | http://purl.obolibrary.org/obo/CHEBI_66919 |
T217 | 998-1007 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T218 | 1147-1149 | Chemical | denotes | RA | http://purl.obolibrary.org/obo/CHEBI_73810 |
T219 | 1200-1209 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T220 | 1337-1339 | Chemical | denotes | IL | http://purl.obolibrary.org/obo/CHEBI_63895|http://purl.obolibrary.org/obo/CHEBI_74072 |
T222 | 1346-1356 | Chemical | denotes | interferon | http://purl.obolibrary.org/obo/CHEBI_52999 |
T223 | 1357-1362 | Chemical | denotes | gamma | http://purl.obolibrary.org/obo/CHEBI_30212 |
T224 | 1521-1524 | Chemical | denotes | CYP | http://purl.obolibrary.org/obo/CHEBI_38559 |
T225 | 1525-1529 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T226 | 1561-1565 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T227 | 1631-1646 | Chemical | denotes | antiviral drugs | http://purl.obolibrary.org/obo/CHEBI_36044 |
T228 | 1631-1640 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T229 | 1641-1646 | Chemical | denotes | drugs | http://purl.obolibrary.org/obo/CHEBI_23888 |
T230 | 1655-1674 | Chemical | denotes | lopinavir/ritonavir | http://purl.obolibrary.org/obo/CHEBI_145924 |
T231 | 1655-1664 | Chemical | denotes | lopinavir | http://purl.obolibrary.org/obo/CHEBI_31781 |
T232 | 1665-1674 | Chemical | denotes | ritonavir | http://purl.obolibrary.org/obo/CHEBI_45409 |
T233 | 1679-1689 | Chemical | denotes | remdesivir | http://purl.obolibrary.org/obo/CHEBI_145994 |
T234 | 1712-1723 | Chemical | denotes | tofacitinib | http://purl.obolibrary.org/obo/CHEBI_71200 |
T235 | 1846-1856 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
T236 | 1880-1882 | Chemical | denotes | RA | http://purl.obolibrary.org/obo/CHEBI_73810 |
T237 | 2124-2135 | Chemical | denotes | ruxolitinib | http://purl.obolibrary.org/obo/CHEBI_66919 |
LitCovid-PD-GO-BP
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T53 | 76-105 | http://purl.obolibrary.org/obo/GO_0006898 | denotes | receptor-mediated endocytosis |
T54 | 94-105 | http://purl.obolibrary.org/obo/GO_0006897 | denotes | endocytosis |
T55 | 135-178 | http://purl.obolibrary.org/obo/GO_2000369 | denotes | regulators of clathrin-mediated endocytosis |
T56 | 149-178 | http://purl.obolibrary.org/obo/GO_0072583 | denotes | clathrin-mediated endocytosis |
T57 | 167-178 | http://purl.obolibrary.org/obo/GO_0006897 | denotes | endocytosis |
T58 | 286-292 | http://purl.obolibrary.org/obo/GO_0016538 | denotes | cyclin |
T59 | 1293-1314 | http://purl.obolibrary.org/obo/GO_0006954 | denotes | inflammatory response |
T60 | 2029-2058 | http://purl.obolibrary.org/obo/GO_0072583 | denotes | clathrin-mediated endocytosis |
T61 | 2047-2058 | http://purl.obolibrary.org/obo/GO_0006897 | denotes | endocytosis |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T147 | 0-111 | Sentence | denotes | As previously described in detail, SARS-CoV-2 enters targeted cells through receptor-mediated endocytosis [12]. |
T148 | 112-325 | Sentence | denotes | Some of the identified regulators of clathrin-mediated endocytosis are members of the numb-associated kinase (NAK) family, such as AP2-associated protein kinase 1 (AAK1) and cyclin G-associated kinase (GAK) [101]. |
T149 | 326-455 | Sentence | denotes | Inhibition of AAK1 may stop the access of the virus into lung cells and also the intracellular assembly of virus particles [102]. |
T150 | 456-536 | Sentence | denotes | Of 47 AAK1 blockers approved for medical use, 6 inhibit AAK1 with high affinity. |
T151 | 537-758 | Sentence | denotes | These include oncologic agents such as erlotinib, sunitinib, ruxolitinib, and fedratinib, which have all been demonstrated to inhibit infection of cells by Dengue virus, Ebola virus, and respiratory syncytial virus [103]. |
T152 | 759-977 | Sentence | denotes | Unfortunately, all these compounds are able to produce adequate NAK inhibition only at doses significantly higher than those normally used in clinical practice and therefore potentially toxic for the patient [104,105]. |
T153 | 978-1174 | Sentence | denotes | Conversely, the JAK inhibitor baricitinib is able to effectively inhibit AAK1 and GAK at the plasma concentration obtained with the approved dosage for the treatment of RA (2 to 4 mg daily) [106]. |
T154 | 1175-1454 | Sentence | denotes | Moreover, as a selective inhibitor of JAK 1 and 2, baricitinib is also able to produce an important dampening of host inflammatory response due to CRS (including IL-6 and interferon gamma) responsible for the more severe forms of interstitial pneumonia during COVID-19 [107,108]. |
T155 | 1455-1696 | Sentence | denotes | Finally, the minimal interaction of baricitinib with the relevant CYP drug-metabolising enzymes makes the drug a possible candidate for inclusion in combination protocols with antiviral drugs such as lopinavir/ritonavir and remdesivir [109]. |
T156 | 1697-1957 | Sentence | denotes | Interestingly, tofacitinib shows no detectable inhibition of AAK1 [104], whereas currently no data are available on the possible effect of other JAK inhibitors approved or tested for RA (such as upadacitinib or filgotinib) in relation to coronavirus infection. |
T157 | 1958-2155 | Sentence | denotes | Unexpectedly, the only clinical trial evaluating the potential role of clathrin-mediated endocytosis blockade in the management of COVID-19 is currently ongoing with ruxolitinib (ChiCTR2000029580). |
LitCovid-PD-HP
Id | Subject | Object | Predicate | Lexical cue | hp_id |
---|---|---|---|---|---|
T83 | 1147-1149 | Phenotype | denotes | RA | http://purl.obolibrary.org/obo/HP_0001370 |
T84 | 1418-1427 | Phenotype | denotes | pneumonia | http://purl.obolibrary.org/obo/HP_0002090 |
T85 | 1880-1882 | Phenotype | denotes | RA | http://purl.obolibrary.org/obo/HP_0001370 |
2_test
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
32205186-28240606-4826922 | 753-756 | 28240606 | denotes | 103 |
32205186-29753658-4826923 | 972-975 | 29753658 | denotes | 105 |
32205186-29545548-4826924 | 1445-1448 | 29545548 | denotes | 107 |
32205186-29649002-4826925 | 1449-1452 | 29649002 | denotes | 108 |