PMC:7600245 / 65551-66788
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T286 | 105-114 | Body_part | denotes | lysosomal | http://purl.org/sig/ont/fma/fma63836 |
T287 | 115-123 | Body_part | denotes | cysteine | http://purl.org/sig/ont/fma/fma82751 |
T288 | 313-317 | Body_part | denotes | skin | http://purl.org/sig/ont/fma/fma7163 |
T289 | 319-324 | Body_part | denotes | liver | http://purl.org/sig/ont/fma/fma7197 |
T290 | 330-334 | Body_part | denotes | lung | http://purl.org/sig/ont/fma/fma7195 |
T291 | 382-390 | Body_part | denotes | cysteine | http://purl.org/sig/ont/fma/fma82751 |
T292 | 661-666 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T293 | 779-783 | Body_part | denotes | cell | http://purl.org/sig/ont/fma/fma68646 |
T294 | 843-847 | Body_part | denotes | lung | http://purl.org/sig/ont/fma/fma7195 |
T295 | 943-948 | Body_part | denotes | lungs | http://purl.org/sig/ont/fma/fma68877 |
LitCovid-PD-UBERON
Id | Subject | Object | Predicate | Lexical cue | uberon_id |
---|---|---|---|---|---|
T30 | 313-317 | Body_part | denotes | skin | http://purl.obolibrary.org/obo/UBERON_0000014 |
T31 | 319-324 | Body_part | denotes | liver | http://purl.obolibrary.org/obo/UBERON_0002107 |
T32 | 330-334 | Body_part | denotes | lung | http://purl.obolibrary.org/obo/UBERON_0002048 |
T33 | 843-847 | Body_part | denotes | lung | http://purl.obolibrary.org/obo/UBERON_0002048 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T309 | 484-492 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T310 | 643-651 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T311 | 748-756 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T312 | 848-854 | Disease | denotes | injury | http://purl.obolibrary.org/obo/MONDO_0021178 |
T313 | 1183-1191 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T662 | 105-114 | http://purl.obolibrary.org/obo/GO_0005764 | denotes | lysosomal |
T663 | 154-162 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T664 | 287-293 | http://purl.obolibrary.org/obo/NCBITaxon_33208 | denotes | animal |
T665 | 313-317 | http://purl.obolibrary.org/obo/UBERON_0000014 | denotes | skin |
T666 | 313-317 | http://purl.obolibrary.org/obo/UBERON_0001003 | denotes | skin |
T667 | 313-317 | http://purl.obolibrary.org/obo/UBERON_0002097 | denotes | skin |
T668 | 313-317 | http://purl.obolibrary.org/obo/UBERON_0002199 | denotes | skin |
T669 | 313-317 | http://www.ebi.ac.uk/efo/EFO_0000962 | denotes | skin |
T670 | 319-324 | http://purl.obolibrary.org/obo/UBERON_0002107 | denotes | liver |
T671 | 319-324 | http://www.ebi.ac.uk/efo/EFO_0000887 | denotes | liver |
T672 | 330-334 | http://purl.obolibrary.org/obo/UBERON_0002048 | denotes | lung |
T673 | 330-334 | http://www.ebi.ac.uk/efo/EFO_0000934 | denotes | lung |
T674 | 520-528 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T675 | 661-666 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T676 | 774-783 | http://purl.obolibrary.org/obo/CLO_0009524 | denotes | Vero cell |
T677 | 826-832 | http://purl.obolibrary.org/obo/NCBITaxon_33208 | denotes | animal |
T678 | 843-847 | http://purl.obolibrary.org/obo/UBERON_0002048 | denotes | lung |
T679 | 843-847 | http://www.ebi.ac.uk/efo/EFO_0000934 | denotes | lung |
T680 | 943-948 | http://www.ebi.ac.uk/efo/EFO_0000934 | denotes | lungs |
T681 | 1024-1034 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activities |
T682 | 1051-1054 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T683 | 1072-1073 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T684 | 1171-1179 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T9195 | 48-56 | Chemical | denotes | molecule | http://purl.obolibrary.org/obo/CHEBI_25367 |
T12773 | 78-87 | Chemical | denotes | inhibitor | http://purl.obolibrary.org/obo/CHEBI_35222 |
T3099 | 115-123 | Chemical | denotes | cysteine | http://purl.obolibrary.org/obo/CHEBI_15356 |
T38887 | 382-390 | Chemical | denotes | cysteine | http://purl.obolibrary.org/obo/CHEBI_15356 |
T92042 | 419-437 | Chemical | denotes | calpain inhibitors | http://purl.obolibrary.org/obo/CHEBI_82824 |
T53518 | 427-437 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
T70302 | 510-519 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T46598 | 690-700 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
T12103 | 927-929 | Chemical | denotes | IL | http://purl.obolibrary.org/obo/CHEBI_63895|http://purl.obolibrary.org/obo/CHEBI_74072 |
T3501 | 992-1001 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T97654 | 1161-1170 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
LitCovid-PD-GO-BP
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T133 | 463-480 | http://purl.obolibrary.org/obo/GO_0019079 | denotes | viral replication |
T134 | 463-480 | http://purl.obolibrary.org/obo/GO_0019058 | denotes | viral replication |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T506 | 0-5 | Sentence | denotes | 4.14. |
T507 | 6-14 | Sentence | denotes | BLD-2660 |
T508 | 15-163 | Sentence | denotes | It an orally bioavailable, small molecule, reversible covalent inhibitor of calpains, non-lysosomal cysteine proteases, with anti-fibrotic activity. |
T509 | 164-335 | Sentence | denotes | BLD-2660 exhibited potent and selective inhibition of calpains 1,2, and 9 and thus was found to be efficacious in multiple animal fibrosis models of skin, liver, and lung. |
T510 | 336-401 | Sentence | denotes | It exhibited high selectivity against related cysteine proteases. |
T511 | 402-505 | Sentence | denotes | Earlier, several calpain inhibitors were found to reduce the viral replication of SARS-CoV-1 [232,233]. |
T512 | 506-677 | Sentence | denotes | The antiviral activity by calpain inhibition was also verified using siRNA to selectively silence expression of the calpain 2 isoform in SARS-CoV infected cells [232,233]. |
T513 | 678-797 | Sentence | denotes | Undisclosed inhibitors by the developing company were found to reduce SARS-CoV-2 replication in Vero cell-based assays. |
T514 | 798-978 | Sentence | denotes | Furthermore, in preclinical animal models of lung injury and fibrosis, BLD-2660 was shown to reduce the expression/production of IL-6 in injured lungs and to reduce fibrosis [234]. |
T515 | 979-1237 | Sentence | denotes | Owing to the antiviral and anti-inflammatory activities of BLD-2660, it has been advanced to a phase 2, randomized, double-blind, placebo-controlled study to evaluate its safety and antiviral activity in COVID-19 hospitalized subjects (NCT04334460; n = 120). |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
2058 | 218-237 | Gene | denotes | calpains 1,2, and 9 | Gene:823 |
2059 | 622-631 | Gene | denotes | calpain 2 | Gene:824 |
2060 | 927-931 | Gene | denotes | IL-6 | Gene:3569 |
2061 | 484-492 | Species | denotes | SARS-CoV | Tax:694009 |
2062 | 748-758 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
2063 | 164-172 | Chemical | denotes | BLD-2660 | |
2064 | 294-302 | Disease | denotes | fibrosis | MESH:D005355 |
2065 | 643-660 | Disease | denotes | SARS-CoV infected | MESH:C000657245 |
2066 | 843-854 | Disease | denotes | lung injury | MESH:D055370 |
2067 | 859-867 | Disease | denotes | fibrosis | MESH:D005355 |
2068 | 963-971 | Disease | denotes | fibrosis | MESH:D005355 |
2069 | 1183-1191 | Disease | denotes | COVID-19 | MESH:C000657245 |