PMC:7600245 / 49590-52711
Annnotations
LitCovid-PD-FMA-UBERON
Id | Subject | Object | Predicate | Lexical cue | fma_id |
---|---|---|---|---|---|
T218 | 35-37 | Body_part | denotes | AG | http://purl.org/sig/ont/fma/fma61898 |
T219 | 169-174 | Body_part | denotes | bowel | http://purl.org/sig/ont/fma/fma7199 |
T220 | 754-764 | Body_part | denotes | pyrimidine | http://purl.org/sig/ont/fma/fma82773 |
T221 | 771-782 | Body_part | denotes | nucleotides | http://purl.org/sig/ont/fma/fma82740 |
T222 | 812-817 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T223 | 850-860 | Body_part | denotes | pyrimidine | http://purl.org/sig/ont/fma/fma82773 |
T224 | 875-880 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T225 | 913-918 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T226 | 1030-1039 | Body_part | denotes | cytokines | http://purl.org/sig/ont/fma/fma84050 |
T227 | 1220-1225 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T228 | 1447-1450 | Body_part | denotes | HIV | http://purl.org/sig/ont/fma/fma278683 |
T229 | 1944-1949 | Body_part | denotes | cells | http://purl.org/sig/ont/fma/fma68646 |
T230 | 2301-2311 | Body_part | denotes | pyrimidine | http://purl.org/sig/ont/fma/fma82773 |
T231 | 2318-2329 | Body_part | denotes | nucleotides | http://purl.org/sig/ont/fma/fma82740 |
T232 | 2731-2734 | Body_part | denotes | HIV | http://purl.org/sig/ont/fma/fma278683 |
T233 | 2748-2752 | Body_part | denotes | foot | http://purl.org/sig/ont/fma/fma9664 |
T234 | 2757-2762 | Body_part | denotes | mouth | http://purl.org/sig/ont/fma/fma49184 |
T235 | 2897-2900 | Body_part | denotes | RNA | http://purl.org/sig/ont/fma/fma67095 |
LitCovid-PD-UBERON
Id | Subject | Object | Predicate | Lexical cue | uberon_id |
---|---|---|---|---|---|
T18 | 2748-2752 | Body_part | denotes | foot | http://purl.obolibrary.org/obo/UBERON_0002387 |
T19 | 2757-2762 | Body_part | denotes | mouth | http://purl.obolibrary.org/obo/UBERON_0000165 |
LitCovid-PD-MONDO
Id | Subject | Object | Predicate | Lexical cue | mondo_id |
---|---|---|---|---|---|
T213 | 156-182 | Disease | denotes | inflammatory bowel disease | http://purl.obolibrary.org/obo/MONDO_0005265 |
T214 | 184-202 | Disease | denotes | multiple sclerosis | http://purl.obolibrary.org/obo/MONDO_0005301 |
T215 | 231-250 | Disease | denotes | autoimmune diseases | http://purl.obolibrary.org/obo/MONDO_0007179 |
T216 | 578-586 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
T217 | 1074-1086 | Disease | denotes | inflammation | http://purl.obolibrary.org/obo/MONDO_0021166 |
T218 | 1296-1305 | Disease | denotes | influenza | http://purl.obolibrary.org/obo/MONDO_0005812 |
T219 | 1419-1428 | Disease | denotes | influenza | http://purl.obolibrary.org/obo/MONDO_0005812 |
T220 | 1523-1531 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T221 | 1613-1621 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T222 | 1671-1679 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T223 | 1857-1865 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T224 | 2706-2715 | Disease | denotes | influenza | http://purl.obolibrary.org/obo/MONDO_0005812 |
T225 | 2748-2770 | Disease | denotes | foot-and-mouth disease | http://purl.obolibrary.org/obo/MONDO_0005765 |
T226 | 2757-2770 | Disease | denotes | mouth disease | http://purl.obolibrary.org/obo/MONDO_0006858 |
T227 | 2920-2928 | Disease | denotes | SARS-CoV | http://purl.obolibrary.org/obo/MONDO_0005091 |
T228 | 3090-3098 | Disease | denotes | COVID-19 | http://purl.obolibrary.org/obo/MONDO_0100096 |
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T493 | 88-89 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T494 | 272-273 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T495 | 404-405 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T496 | 787-796 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activated |
T497 | 797-798 | http://purl.obolibrary.org/obo/CLO_0001021 | denotes | B |
T498 | 812-817 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T499 | 875-880 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T500 | 913-918 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T501 | 1165-1166 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T502 | 1198-1201 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T503 | 1220-1225 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T504 | 1266-1273 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | viruses |
T505 | 1306-1311 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T506 | 1342-1350 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T507 | 1351-1354 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T508 | 1429-1430 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | A |
T509 | 1431-1436 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T510 | 1466-1469 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T511 | 1506-1514 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T512 | 1682-1690 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T513 | 1840-1848 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T514 | 1927-1936 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activated |
T515 | 1944-1949 | http://purl.obolibrary.org/obo/GO_0005623 | denotes | cells |
T516 | 2022-2027 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T517 | 2122-2123 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T518 | 2513-2521 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T519 | 2584-2587 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T520 | 2662-2663 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T521 | 2689-2697 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T522 | 2716-2723 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | viruses |
T523 | 2725-2728 | http://purl.obolibrary.org/obo/CLO_0001002 | denotes | 162 |
T524 | 2738-2741 | http://purl.obolibrary.org/obo/CLO_0001003 | denotes | 163 |
T525 | 2757-2762 | http://www.ebi.ac.uk/efo/EFO_0000825 | denotes | mouth |
T526 | 2771-2776 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | virus |
T527 | 2793-2794 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T528 | 2818-2821 | http://purl.obolibrary.org/obo/CLO_0051582 | denotes | has |
T529 | 2837-2845 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
T530 | 2901-2908 | http://purl.obolibrary.org/obo/NCBITaxon_10239 | denotes | viruses |
T531 | 2980-2981 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T532 | 2999-3004 | http://purl.obolibrary.org/obo/CLO_0007225 | denotes | label |
T533 | 3053-3061 | http://purl.obolibrary.org/obo/CLO_0001658 | denotes | activity |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T714 | 18-25 | Chemical | denotes | Calcium | http://purl.obolibrary.org/obo/CHEBI_22984 |
T715 | 35-37 | Chemical | denotes | AG | http://purl.obolibrary.org/obo/CHEBI_27569|http://purl.obolibrary.org/obo/CHEBI_40618|http://purl.obolibrary.org/obo/CHEBI_73757 |
T25593 | 106-114 | Chemical | denotes | molecule | http://purl.obolibrary.org/obo/CHEBI_25367 |
T7933 | 274-282 | Chemical | denotes | biphenyl | http://purl.obolibrary.org/obo/CHEBI_17097 |
T40831 | 283-292 | Chemical | denotes | carbamoyl | http://purl.obolibrary.org/obo/CHEBI_23004|http://purl.obolibrary.org/obo/CHEBI_33100 |
T2210 | 293-305 | Chemical | denotes | cyclopentene | http://purl.obolibrary.org/obo/CHEBI_49155 |
T4722 | 646-650 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T60213 | 672-686 | Chemical | denotes | dihydroorotate | http://purl.obolibrary.org/obo/CHEBI_30867 |
T49164 | 754-764 | Chemical | denotes | pyrimidine | http://purl.obolibrary.org/obo/CHEBI_16898 |
T10698 | 771-782 | Chemical | denotes | nucleotides | http://purl.obolibrary.org/obo/CHEBI_36976 |
T11341 | 850-860 | Chemical | denotes | pyrimidine | http://purl.obolibrary.org/obo/CHEBI_16898 |
T90920 | 1043-1045 | Chemical | denotes | IL | http://purl.obolibrary.org/obo/CHEBI_63895|http://purl.obolibrary.org/obo/CHEBI_74072 |
T57301 | 1109-1123 | Chemical | denotes | dihydroorotate | http://purl.obolibrary.org/obo/CHEBI_30867 |
T89861 | 1174-1183 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T67353 | 1332-1341 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T28939 | 1496-1505 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T27522 | 1830-1839 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T48024 | 2141-2149 | Chemical | denotes | molecule | http://purl.obolibrary.org/obo/CHEBI_25367 |
T51342 | 2155-2164 | Chemical | denotes | quinoline | http://purl.obolibrary.org/obo/CHEBI_17362 |
T32891 | 2165-2180 | Chemical | denotes | carboxylic acid | http://purl.obolibrary.org/obo/CHEBI_33575 |
T41022 | 2176-2180 | Chemical | denotes | acid | http://purl.obolibrary.org/obo/CHEBI_37527 |
T40724 | 2222-2236 | Chemical | denotes | dihydroorotate | http://purl.obolibrary.org/obo/CHEBI_30867 |
T19589 | 2301-2311 | Chemical | denotes | pyrimidine | http://purl.obolibrary.org/obo/CHEBI_16898 |
T32360 | 2318-2329 | Chemical | denotes | nucleotides | http://purl.obolibrary.org/obo/CHEBI_36976 |
T11825 | 2432-2446 | Chemical | denotes | antineoplastic | http://purl.obolibrary.org/obo/CHEBI_35610 |
T78103 | 2531-2552 | Chemical | denotes | antineoplastic agents | http://purl.obolibrary.org/obo/CHEBI_35610 |
T86303 | 2579-2583 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T36415 | 2648-2652 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T14871 | 2679-2688 | Chemical | denotes | antiviral | http://purl.obolibrary.org/obo/CHEBI_22587 |
T73829 | 2849-2888 | Chemical | denotes | dihydroorotate dehydrogenase inhibitors | http://purl.obolibrary.org/obo/CHEBI_68542 |
T76979 | 2849-2863 | Chemical | denotes | dihydroorotate | http://purl.obolibrary.org/obo/CHEBI_30867 |
T66976 | 2878-2888 | Chemical | denotes | inhibitors | http://purl.obolibrary.org/obo/CHEBI_35222 |
T64357 | 2953-2957 | Chemical | denotes | drug | http://purl.obolibrary.org/obo/CHEBI_23888 |
T82803 | 2999-3004 | Chemical | denotes | label | http://purl.obolibrary.org/obo/CHEBI_35209 |
LitCovid-PD-GO-BP
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T84 | 738-750 | http://purl.obolibrary.org/obo/GO_0009058 | denotes | biosynthesis |
T85 | 1074-1086 | http://purl.obolibrary.org/obo/GO_0006954 | denotes | inflammation |
T86 | 2285-2297 | http://purl.obolibrary.org/obo/GO_0009058 | denotes | biosynthesis |
LitCovid-PD-HP
Id | Subject | Object | Predicate | Lexical cue | hp_id |
---|---|---|---|---|---|
T48 | 156-182 | Phenotype | denotes | inflammatory bowel disease | http://purl.obolibrary.org/obo/HP_0002037 |
T49 | 231-250 | Phenotype | denotes | autoimmune diseases | http://purl.obolibrary.org/obo/HP_0002960 |
T50 | 1252-1257 | Phenotype | denotes | fever | http://purl.obolibrary.org/obo/HP_0001945 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T369 | 0-4 | Sentence | denotes | 4.4. |
T370 | 5-71 | Sentence | denotes | Vidofludimus Calcium (Immunic AG, IMU-838) and Brequinar (DuP-785) |
T371 | 72-265 | Sentence | denotes | Vidofludimus is a synthetic small molecule that is under investigation for treating inflammatory bowel disease, multiple sclerosis, and other inflammatory and autoimmune diseases [154,155,156]. |
T372 | 266-392 | Sentence | denotes | It is a biphenyl-carbamoyl-cyclopentene derivative (Figure 7) that is being developed as oral formulation for therapeutic use. |
T373 | 393-625 | Sentence | denotes | Currently, a prospective, randomized, multi-center, double-blinded, and placebo-controlled study is ongoing to evaluate the safety and efficacy of vidofludimus as an adjunct therapy in COVID-19 patients (NCT04379271; n = 230) [157]. |
T374 | 626-818 | Sentence | denotes | The investigational drug selectively inhibits dihydroorotate dehydrogenase, an important enzyme for the de novo biosynthesis of pyrimidine-based nucleotides, in activated B and T immune cells. |
T375 | 819-939 | Sentence | denotes | Such inhibition diminishes the pyrimidine pool in these cells, which subsequently exposes the cells to metabolic stress. |
T376 | 940-1093 | Sentence | denotes | It also diminishes the release of T helper 1 (Th1) and T helper 17 (Th17) proinflammatory cytokines of IL-17 and IFN-γ, which reduces inflammation [154]. |
T377 | 1094-1312 | Sentence | denotes | Interestingly, dihydroorotate dehydrogenase inhibition also results in a direct antiviral effect, which has been exhibited in cells infected with hemorrhagic fever-causing viruses, cytomegalovirus, and influenza virus. |
T378 | 1313-1457 | Sentence | denotes | In fact, IMU-838′s antiviral activity has been demonstrated in vitro against arenavirus, cytomegalovirus, influenza A virus, HCV, and HIV [157]. |
T379 | 1458-1540 | Sentence | denotes | IMU-838 has also effectively promoted antiviral activity against SARS-CoV-2 [157]. |
T380 | 1541-1624 | Sentence | denotes | Specifically, IMU-838 inhibited the replication of clinical isolates of SARS-CoV-2. |
T381 | 1625-1810 | Sentence | denotes | In cellular assays, IMU-838 promoted the anti-SARS-CoV-2 activity at concentrations lower than those that have been considered in previous and ongoing clinical trials [154,155,156,157]. |
T382 | 1811-2098 | Sentence | denotes | Overall, IMU-838′s antiviral activity against SARS-CoV-2 as well as its selective immunomodulatory effect targeting activated immune cells appear to be interesting, particularly that it potentially prevents the virus reactivation that may happen with other immunomodulatory agents [157]. |
T383 | 2099-2251 | Sentence | denotes | Likewise, brequinar is a synthetic, small molecule, and quinoline-carboxylic acid derivative (Figure 7) that also inhibits dihydroorotate dehydrogenase. |
T384 | 2252-2340 | Sentence | denotes | It eventually blocks the de novo biosynthesis of pyrimidine-based nucleotides [158,159]. |
T385 | 2341-2400 | Sentence | denotes | Accordingly, brequinar possesses immunosuppressive effects. |
T386 | 2401-2559 | Sentence | denotes | Furthermore, it also possesses antineoplastic properties that can be exploited to enhance the in vivo antitumor activity of other antineoplastic agents [160]. |
T387 | 2560-2625 | Sentence | denotes | Alternatively, the drug has also antiparasitic effects [160,161]. |
T388 | 2626-2783 | Sentence | denotes | More importantly, the drug exhibits a broad-spectrum antiviral activity against influenza viruses [162], HIV-1 [163], and foot-and-mouth disease virus [164]. |
T389 | 2784-2937 | Sentence | denotes | In fact, a pre-print under review has documented the activity of dihydroorotate dehydrogenase inhibitors against RNA viruses, including SARS-CoV-2 [165]. |
T390 | 2938-3121 | Sentence | denotes | Currently, the drug is being evaluated in a randomized, open-label trial to assess its safety and anti-coronavirus activity in hospitalized adults with COVID-19 (NCT04425252; n = 24). |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
1556 | 5-25 | Chemical | denotes | Vidofludimus Calcium | |
1557 | 39-46 | Chemical | denotes | IMU-838 | MESH:C553728 |
1566 | 587-595 | Species | denotes | patients | Tax:9606 |
1567 | 72-84 | Chemical | denotes | Vidofludimus | MESH:C553728 |
1568 | 274-305 | Chemical | denotes | biphenyl-carbamoyl-cyclopentene | |
1569 | 540-552 | Chemical | denotes | vidofludimus | MESH:C553728 |
1570 | 156-182 | Disease | denotes | inflammatory bowel disease | MESH:D015212 |
1571 | 184-202 | Disease | denotes | multiple sclerosis | MESH:D009103 |
1572 | 231-250 | Disease | denotes | autoimmune diseases | MESH:D001327 |
1573 | 578-586 | Disease | denotes | COVID-19 | MESH:C000657245 |
1594 | 672-700 | Gene | denotes | dihydroorotate dehydrogenase | Gene:1723 |
1595 | 1043-1048 | Gene | denotes | IL-17 | Gene:3605 |
1596 | 1053-1058 | Gene | denotes | IFN-γ | Gene:3458 |
1597 | 1109-1137 | Gene | denotes | dihydroorotate dehydrogenase | Gene:1723 |
1598 | 1296-1311 | Species | denotes | influenza virus | Tax:11308 |
1599 | 1419-1436 | Species | denotes | influenza A virus | Tax:11320 |
1600 | 1523-1533 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
1601 | 1613-1623 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
1602 | 1857-1867 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
1603 | 1671-1681 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
1604 | 754-770 | Chemical | denotes | pyrimidine-based | |
1605 | 850-860 | Chemical | denotes | pyrimidine | MESH:C030986 |
1606 | 1322-1329 | Chemical | denotes | IMU-838 | MESH:C553728 |
1607 | 1458-1465 | Chemical | denotes | IMU-838 | MESH:C553728 |
1608 | 1555-1562 | Chemical | denotes | IMU-838 | MESH:C553728 |
1609 | 1645-1652 | Chemical | denotes | IMU-838 | MESH:C553728 |
1610 | 1820-1827 | Chemical | denotes | IMU-838 | MESH:C553728 |
1611 | 1074-1086 | Disease | denotes | inflammation | MESH:D007249 |
1612 | 1226-1234 | Disease | denotes | infected | MESH:D007239 |
1613 | 1240-1257 | Disease | denotes | hemorrhagic fever | MESH:D006480 |
1624 | 2222-2250 | Gene | denotes | dihydroorotate dehydrogenase | Gene:1723 |
1625 | 2849-2877 | Gene | denotes | dihydroorotate dehydrogenase | Gene:1723 |
1626 | 2706-2723 | Species | denotes | influenza viruses | Tax:11308 |
1627 | 2731-2736 | Species | denotes | HIV-1 | Tax:11676 |
1628 | 2748-2776 | Species | denotes | foot-and-mouth disease virus | Tax:12110 |
1629 | 2920-2930 | Species | denotes | SARS-CoV-2 | Tax:2697049 |
1630 | 3041-3052 | Species | denotes | coronavirus | Tax:11118 |
1631 | 2155-2180 | Chemical | denotes | quinoline-carboxylic acid | |
1632 | 2301-2329 | Chemical | denotes | pyrimidine-based nucleotides | |
1633 | 3090-3098 | Disease | denotes | COVID-19 | MESH:C000657245 |