PMC:7571312 / 94806-95846
Annnotations
LitCovid-PD-CLO
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T659 | 385-386 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T660 | 541-542 | http://purl.obolibrary.org/obo/CLO_0001020 | denotes | a |
T661 | 931-933 | http://purl.obolibrary.org/obo/CLO_0007874 | denotes | MS |
T662 | 968-973 | http://purl.obolibrary.org/obo/CLO_0007706 | denotes | M + H |
LitCovid-PD-CHEBI
Id | Subject | Object | Predicate | Lexical cue | chebi_id |
---|---|---|---|---|---|
T1836 | 77-83 | Chemical | denotes | chloro | http://purl.obolibrary.org/obo/CHEBI_47853 |
T1837 | 86-89 | Chemical | denotes | oxo | http://purl.obolibrary.org/obo/CHEBI_46629 |
T1838 | 120-126 | Chemical | denotes | methyl | http://purl.obolibrary.org/obo/CHEBI_32875|http://purl.obolibrary.org/obo/CHEBI_29309 |
T1840 | 127-133 | Chemical | denotes | propyl | http://purl.obolibrary.org/obo/CHEBI_26308 |
T1841 | 134-139 | Chemical | denotes | amino | http://purl.obolibrary.org/obo/CHEBI_46882 |
T1842 | 140-148 | Chemical | denotes | carbonyl | http://purl.obolibrary.org/obo/CHEBI_23019 |
T1843 | 150-163 | Chemical | denotes | 3-methylbutyl | http://purl.obolibrary.org/obo/CHEBI_30359 |
T1844 | 167-174 | Chemical | denotes | methoxy | http://purl.obolibrary.org/obo/CHEBI_32772|http://purl.obolibrary.org/obo/CHEBI_44520 |
T1846 | 175-184 | Chemical | denotes | 1H-indole | http://purl.obolibrary.org/obo/CHEBI_16881 |
T1847 | 175-177 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1848 | 178-184 | Chemical | denotes | indole | http://purl.obolibrary.org/obo/CHEBI_35581 |
T1849 | 187-198 | Chemical | denotes | carboxamide | http://purl.obolibrary.org/obo/CHEBI_23004|http://purl.obolibrary.org/obo/CHEBI_37622 |
T1851 | 216-218 | Chemical | denotes | N2 | http://purl.obolibrary.org/obo/CHEBI_17997 |
T1852 | 220-239 | Chemical | denotes | tert-butoxycarbonyl | http://purl.obolibrary.org/obo/CHEBI_48502 |
T1853 | 252-258 | Chemical | denotes | chloro | http://purl.obolibrary.org/obo/CHEBI_47853 |
T1854 | 261-264 | Chemical | denotes | oxo | http://purl.obolibrary.org/obo/CHEBI_46629 |
T1855 | 295-301 | Chemical | denotes | methyl | http://purl.obolibrary.org/obo/CHEBI_32875|http://purl.obolibrary.org/obo/CHEBI_29309 |
T1857 | 302-308 | Chemical | denotes | propyl | http://purl.obolibrary.org/obo/CHEBI_26308 |
T1858 | 312-318 | Chemical | denotes | methyl | http://purl.obolibrary.org/obo/CHEBI_32875|http://purl.obolibrary.org/obo/CHEBI_29309 |
T1860 | 472-480 | Chemical | denotes | methanol | http://purl.obolibrary.org/obo/CHEBI_17790 |
T1861 | 481-491 | Chemical | denotes | chloroform | http://purl.obolibrary.org/obo/CHEBI_35255 |
T1862 | 556-558 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1863 | 564-568 | Chemical | denotes | DMSO | http://purl.obolibrary.org/obo/CHEBI_28262 |
T1864 | 585-587 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1865 | 609-611 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1866 | 633-635 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1867 | 647-649 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1868 | 661-663 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1869 | 685-687 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1870 | 709-711 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1871 | 733-735 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1872 | 761-763 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1873 | 775-777 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1874 | 817-819 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1875 | 831-833 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1876 | 845-847 | Chemical | denotes | 1H | http://purl.obolibrary.org/obo/CHEBI_49637 |
T1877 | 931-933 | Chemical | denotes | MS | http://purl.obolibrary.org/obo/CHEBI_73613 |
LitCovid-sentences
Id | Subject | Object | Predicate | Lexical cue |
---|---|---|---|---|
T543 | 0-405 | Sentence | denotes | Following the procedure described for the preparation of N-((1S)-1-{[((1S)-3-chloro-2-oxo-1-{[(3S)-2-oxopyrrolidin-3-yl]methyl}propyl)amino]carbonyl}-3-methylbutyl)-4-methoxy-1H-indole-2-carboxamide but substituting N2-(tert-butoxycarbonyl)-N1-((1S)-3-chloro-2-oxo-1-{[(3S)-2-oxopyrrolidin-3-yl]methyl}propyl)-5-methyl-l-norleucinamide and making no other critical variations provided a crude yellow foam. |
T544 | 406-555 | Sentence | denotes | This material was purified by Biotage MPLC (25 M column, 2.5–3.5% methanol/chloroform) to afford 307 mg (73%) of the title compound as a white solid. |
T545 | 556-1040 | Sentence | denotes | 1H NMR (DMSO-d6) δ 11.57 (s, 1H), 8.59 (d, J = 8 Hz, 1H), 8.41 (d, J = 4 Hz, 1H), 7.64 (s, 1H), 7.37 (s, 1H), 7.09 (t, J = 8 Hz, 1H), 7.00 (d, J = 8 Hz, 1H), 6.49 (d, J = 8 Hz, 1H), 4.59 (s, 2H), 4.44 (m, 1H), 4.35 (m, 1H), 3.87 (s, 3H), 3.08 (m, 2H), 2.26 (m, 1H), 2.07 (m, 1H), 1.98 (m, 1H), 1.70–1.51 (m, 5H), 1.25 (m, 2H), 0.88 (d, J = 4 Hz, 3H), 0.86 (d, J = 4 Hz, 3H); MS (ESI+) for C25H33ClN4O5m/z 505.2 (M + H)+; HRMS (ESI+) calcd for C25H33ClN4O5+H1 505.2212, found 505.2204. |
LitCovid-PubTator
Id | Subject | Object | Predicate | Lexical cue | tao:has_database_id |
---|---|---|---|---|---|
1838 | 1009-1014 | Species | denotes | O5+H1 | Tax:2491878 |
1839 | 472-480 | Chemical | denotes | methanol | MESH:D000432 |
1840 | 481-491 | Chemical | denotes | chloroform | MESH:D002725 |
1841 | 977-981 | Disease | denotes | HRMS |